SCHEMBL5206192

SCHEMBL5206192

CC(C)(C)OC(=O)NCc1ccc(Oc2ccccc2N(Cc2ccc(-c3ccccc3)cc2)C(=O)CCC(=O)NCc2ccccc2F)cc1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.40
ALDH1A1 P00352 3/20 0.39
SDCBP O00560 1/20 0.38
SDC2 P34741 1/20 0.38
LPAR1 Q92633 3/20 0.38
LPAR5 Q9H1C0 3/20 0.38
TDP1 Q9NUW8 1/20 0.38
TSPO P30536 1/20 0.38
KMT2A Q03164 3/20 0.37
PTPN1 P18031 1/20 0.37
HTT P42858 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
MEN1 O00255 2/20 0.36
FAAH O00519 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5204311 0.93 ALDH1A1 (0.42) HDAC1ALDH1A1SDCBPSDC2LPAR1
SCHEMBL5202464 0.88 ALDH1A1 (0.41) HDAC1ALDH1A1TSPOPTPN1HTT
SCHEMBL5204889 0.88 HDAC1 (0.47) HDAC1ALDH1A1SDCBPSDC2TSPO
SCHEMBL5204997 0.87 ALDH1A1 (0.43) HDAC1ALDH1A1LPAR1LPAR5TSPO
SCHEMBL5206214 0.86 ALDH1A1 (0.40) HDAC1ALDH1A1SDCBPSDC2KMT2A
Hydrochloric Acid SCHEMBL5205960 0.86 LPAR1 (0.41) ALDH1A1LPAR1LPAR5TSPOKMT2A
SCHEMBL5203418 0.85 ALDH1A1 (0.40) HDAC1ALDH1A1SDCBPSDC2TSPO
SCHEMBL5204960 0.81 HTT (0.37) ALDH1A1TSPOKMT2AHTTSMN1; SMN2
SCHEMBL5208000 0.80 HDAC1 (0.44) HDAC1SDCBPSDC2TDP1TSPO
Hydrochloric Acid SCHEMBL5203571 0.80 SSTR5 (0.43) ALDH1A1LPAR1LPAR5TSPOKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160887-B1 Aromatic amine derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-09 US disclosed
EP-1123918-B1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME TAKEDA PHARMACEUTICAL (JP) 2005-03-09 EP disclosed
EP-1123918-A1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME Takeda Chemical Industries, Ltd. (JP) 2001-08-16 EP disclosed