SCHEMBL5202596

SCHEMBL5202596

N#Cc1cccc(Cn2cc(C3CCN(C(=O)c4ccc5c(c4)OCO5)C3)c3ccccc32)c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
TSHR P16473 1/20 0.47
SLC2A1 P11166 1/20 0.47
IGF2BP1 Q9NZI8 1/20 0.46
LMNA P02545 2/20 0.45
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
HTR2B P41595 1/20 0.44
SMO Q99835 1/20 0.43
HRH2 P25021 3/20 0.42
POLB P06746 1/20 0.41
KDM4E B2RXH2 1/20 0.41
HSD11B1 P28845 1/20 0.41
KDM1A O60341 1/20 0.41
PAX8 Q06710 1/20 0.40
MCHR1 Q99705 1/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13445248 0.81 SMO (0.57) SLC2A1HTR2AHTR2CHTR2BSMO
SCHEMBL5201634 0.79 SLC2A1 (0.47) ALDH1A1SLC2A1LMNAHTR2AHTR2C
SCHEMBL4859724 0.79 SMO (0.46) ALDH1A1SLC2A1LMNAHTR2AHTR2C
SCHEMBL5202604 0.79 SLC2A1 (0.46) SLC2A1HTR2AHTR2CHTR2BSMO
SCHEMBL4861849 0.78 KDM1A (0.46) ALDH1A1SLC2A1LMNAHTR2AHTR2C
SCHEMBL5203146 0.78 SMO (0.47) ALDH1A1SLC2A1LMNAHTR2AHTR2C
SCHEMBL5202216 0.77 SMO (0.49) ALDH1A1SLC2A1LMNAHTR2AHTR2C
SCHEMBL3599338 0.77 SLC2A1 (0.55) ALDH1A1TSHRSLC2A1HTR2AHTR2C
SCHEMBL4853409 0.75 SLC2A1 (0.50) ALDH1A1SLC2A1LMNAHTR2AHTR2C
SCHEMBL5206911 0.73 SLC2A1 (0.57) ALDH1A1TSHRSLC2A1LMNAHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP disclosed