SCHEMBL5202604

SCHEMBL5202604

N#Cc1cccc(Cn2cc(C3CCN(C(=O)C4=COC(Cc5ccccc5)O4)C3)c3ccccc32)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.46
SMO Q99835 1/20 0.44
HTR2A P28223 3/20 0.43
HTR2C P28335 3/20 0.43
HTR2B P41595 3/20 0.43
HRH2 P25021 5/20 0.41
KDM1A O60341 1/20 0.40
MGLL Q99685 1/20 0.38
DRD2 P14416 1/20 0.37
HTR6 P50406 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.37
SIRT1 Q96EB6 1/20 0.37
CCR3 P51677 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PIK3CA P42336 1/20 0.36
MTOR P42345 1/20 0.36
CFD P00746 1/20 0.36
CNR2 P34972 1/20 0.36
SLC5A1 P13866 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5202596 0.79 ALDH1A1 (0.47) SLC2A1SMOHTR2AHTR2CHTR2B
SCHEMBL5201634 0.78 SLC2A1 (0.47) SLC2A1SMOHTR2AHTR2CHTR2B
SCHEMBL4859724 0.78 SMO (0.46) SLC2A1SMOHTR2AHTR2CHTR2B
SCHEMBL5202216 0.78 SMO (0.49) SLC2A1SMOHTR2AHTR2CHTR2B
SCHEMBL4861849 0.77 KDM1A (0.46) SLC2A1SMOHTR2AHTR2CHTR2B
SCHEMBL13445248 0.77 SMO (0.57) SLC2A1SMOHTR2AHTR2CHTR2B
SCHEMBL3599338 0.71 SLC2A1 (0.55) SLC2A1SMOHTR2AHTR2CHTR2B
SCHEMBL5203146 0.70 SMO (0.47) SLC2A1SMOHTR2AHTR2CHTR2B
SCHEMBL5205834 0.69 SMO (0.48) SLC2A1SMOHTR2AHTR2CHTR2B
SCHEMBL5206733 0.69 SCD5 (0.47) SLC2A1SMOHTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP disclosed