SCHEMBL5202930

SCHEMBL5202930

O=C(Cc1ccc(Cl)cc1)N1CCC(c2cn(Cc3cccc(F)c3)c3ccccc23)C1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.59
ALDH1A1 P00352 8/20 0.53
LMNA P02545 7/20 0.53
NPSR1 Q6W5P4 3/20 0.53
HTT P42858 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.51
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
TSHR P16473 1/20 0.49
TDP1 Q9NUW8 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.45
HRH2 P25021 1/20 0.45
CNR2 P34972 1/20 0.44
POLB P06746 1/20 0.44
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
HTR2B P41595 1/20 0.44
SLC5A1 P13866 1/20 0.44
SLC5A2 P31639 1/20 0.44
TP53 P04637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5204486 0.87 MAPT (0.54) SLC2A1ALDH1A1LMNANPSR1HTT
SCHEMBL5818040 0.87 SLC2A1 (0.47) SLC2A1ALDH1A1LMNANPSR1HTT
SCHEMBL4859827 0.85 SLC2A1 (0.61) SLC2A1ALDH1A1LMNANPSR1HTT
SCHEMBL14181452 0.80 SLC2A1 (0.57) SLC2A1ALDH1A1LMNANPSR1HTT
SCHEMBL5203232 0.80 LMNA (0.51) ALDH1A1LMNANPSR1HTTPOLB
SCHEMBL5206324 0.80 SLC2A1 (0.50) SLC2A1ALDH1A1LMNANPSR1HTT
SCHEMBL5201638 0.79 SLC2A1 (0.49) SLC2A1ALDH1A1LMNANPSR1HTT
SCHEMBL4859500 0.79 KMT2A (0.52) ALDH1A1LMNANPSR1HTTSMN1; SMN2
SCHEMBL4859525 0.78 SLC2A1 (0.63) SLC2A1ALDH1A1LMNANPSR1HTT
SCHEMBL3615414 0.77 SLC2A1 (0.64) SLC2A1ALDH1A1LMNANPSR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP disclosed