SCHEMBL5202941

SCHEMBL5202941

CCOc1cc(C2=NN(C(=O)c3cccc([N+](=O)[O-])c3)CCC2)ccc1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 6/20 0.51
HTT P42858 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
NCOA1 Q15788 1/20 0.47
NCOA3 Q9Y6Q9 1/20 0.47
ALDH1A1 P00352 3/20 0.46
LMNA P02545 3/20 0.46
NPSR1 Q6W5P4 2/20 0.46
PKM P14618 1/20 0.46
MAOB P27338 1/20 0.45
POLB P06746 1/20 0.44
GRIN2C Q14957 1/20 0.44
MAPT P10636 3/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
SETD7 Q8WTS6 1/20 0.42
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3919528 0.96 PGR (0.53) PGRHTTSMN1; SMN2NCOA1NCOA3
SCHEMBL6583356 0.92 SETD7 (0.52) PGRSMN1; SMN2ALDH1A1POLBMAPT
SCHEMBL5203350 0.90 PGR (0.63) PGRHTTSMN1; SMN2ALDH1A1LMNA
SCHEMBL6583496 0.90 SETD7 (0.51) PGRHTTALDH1A1LMNAPOLB
SCHEMBL6582141 0.90 SETD7 (0.51) PGRHTTSMN1; SMN2ALDH1A1POLB
SCHEMBL6581955 0.89 SETD7 (0.52) PGRHTTSMN1; SMN2ALDH1A1POLB
SCHEMBL6583352 0.88 PGR (0.50) PGRSMN1; SMN2ALDH1A1LMNANPSR1
SCHEMBL6584768 0.87 KMT2A (0.49) PGRHTTSMN1; SMN2ALDH1A1POLB
SCHEMBL6579233 0.86 PGR (0.49) PGRSMN1; SMN2ALDH1A1LMNAPOLB
SCHEMBL5202716 0.86 ALDH1A1 (0.49) PGRSMN1; SMN2ALDH1A1LMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1087946-B1 ARYL ALKANOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2007-01-10 EP disclosed
US-6417188-B1 ENZYME INHIBITORS OF PHOSPHODIESTERASE MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 2002-07-09 US disclosed