SCHEMBL5203350

SCHEMBL5203350

CCOc1cc(C2=NN(C(=O)c3ccc([N+](=O)[O-])cc3)CCC2)ccc1OC

nearest known ligand 0.63

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PGR P06401 10/20 0.63
ALDH1A1 P00352 3/20 0.48
POLB P06746 2/20 0.48
MAOB P27338 1/20 0.47
MAPT P10636 4/20 0.45
LMNA P02545 2/20 0.45
MAPK1 P28482 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
GAA P10253 1/20 0.45
HTT P42858 1/20 0.44
HPGD P15428 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
PDE4B Q07343 2/20 0.42
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6578966 0.93 PGR (0.55) PGRALDH1A1POLBMAPTLMNA
SCHEMBL6606027 0.93 PGR (0.70) PGRALDH1A1POLBMAOBMAPT
SCHEMBL5202941 0.90 PGR (0.51) PGRALDH1A1POLBMAOBMAPT
SCHEMBL6583352 0.88 PGR (0.50) PGRALDH1A1POLBMAPTLMNA
SCHEMBL6584769 0.88 PGR (0.50) PGRALDH1A1POLBMAPTLMNA
SCHEMBL13210796 0.88 ALDH1A1 (0.53) PGRALDH1A1POLBMAOBMAPT
SCHEMBL6584768 0.88 KMT2A (0.49) PGRALDH1A1POLBMAPTHTT
SCHEMBL6579233 0.87 PGR (0.49) PGRALDH1A1POLBMAPTLMNA
SCHEMBL3920897 0.87 ALDH1A1 (0.52) PGRALDH1A1POLBMAOBMAPT
SCHEMBL6583496 0.86 SETD7 (0.51) PGRALDH1A1POLBMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1087946-B1 ARYL ALKANOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2007-01-10 EP disclosed
US-6417188-B1 ENZYME INHIBITORS OF PHOSPHODIESTERASE MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 2002-07-09 US disclosed