SCHEMBL5203370

SCHEMBL5203370

COc1cccc(Cn2cc(C3CCN(C(=O)CC(C)(C)C)C3)c3ccccc32)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH2 P25021 5/20 0.47
MAPT P10636 1/20 0.46
HTR2A P28223 5/20 0.45
HTR2C P28335 5/20 0.45
HTR2B P41595 5/20 0.45
SLC2A1 P11166 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
HTT P42858 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
POLB P06746 1/20 0.44
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
NCOR2 Q9Y618 1/20 0.43
SLC5A1 P13866 1/20 0.42
SLC5A2 P31639 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4852934 0.90 HRH2 (0.50) HRH2MAPTHTR2AHTR2CHTR2B
SCHEMBL5205779 0.88 HRH2 (0.49) HRH2MAPTHTR2AHTR2CHTR2B
SCHEMBL5204486 0.86 MAPT (0.54) HRH2MAPTHTR2AHTR2CHTR2B
SCHEMBL4857604 0.84 MAPT (0.53) HRH2MAPTHTR2AHTR2CHTR2B
SCHEMBL5202293 0.84 THRB (0.49) HRH2MAPTHTR2AHTR2CHTR2B
SCHEMBL4859761 0.83 HRH2 (0.48) HRH2MAPTHTR2AHTR2CHTR2B
SCHEMBL5202181 0.81 HRH2 (0.49) HRH2MAPTHTR2AHTR2CHTR2B
SCHEMBL5203382 0.80 MAPT (0.46) HRH2MAPTHTR2AHTR2CHTR2B
SCHEMBL5204484 0.80 SLC2A1 (0.47) HRH2MAPTHTR2AHTR2CHTR2B
SCHEMBL4858356 0.80 CREBBP (0.42) HRH2ALDH1A1POLBHDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP disclosed