SCHEMBL5203497

SCHEMBL5203497

COc1cc(OB(O)O)cc(OC)c1OCC(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.35
CYP1A2 P05177 2/20 0.35
ALDH1A1 P00352 3/20 0.35
MAPT P10636 3/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
KDM4E B2RXH2 2/20 0.35
USP2 O75604 1/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
THRB P10828 1/20 0.35
G6PD P11413 1/20 0.35
ALOX15 P16050 1/20 0.35
CASP1 P29466 1/20 0.35
HSD17B10 Q99714 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CYP2C19 P33261 2/20 0.34
CYP3A4 P08684 2/20 0.34
MRGPRX4 Q96LA9 1/20 0.34
TUBB4A P04350 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6339479 0.81 MAPT (0.37) CYP2C9CYP1A2ALDH1A1MAPTMEN1
SCHEMBL5205549 0.80 HTR2A (0.49) CYP1A2ALDH1A1MAPTKDM4ECYP2C19
SCHEMBL5203576 0.78 TNFRSF1A (0.45) ALDH1A1MAPTMEN1KMT2AL3MBTL1
SCHEMBL5208220 0.78 SMN1; SMN2 (0.48) ALDH1A1MAPTMEN1KMT2AL3MBTL1
SCHEMBL5207796 0.77 CYP3A4 (0.52) CYP1A2MAPTMEN1KMT2ACYP3A4
SCHEMBL5203586 0.75 MAPT (0.40) CYP2C9CYP1A2ALDH1A1MAPTMEN1
Hydrochloric Acid SCHEMBL5205490 0.73 MAPT (0.52) CYP2C9CYP1A2ALDH1A1MAPTMEN1
SCHEMBL5205202 0.73 TPMT (0.54) ALDH1A1MEN1KMT2AHSD17B10L3MBTL1
SCHEMBL5203822 0.73 GAA (0.48) ALDH1A1MAPTMEN1KMT2AKDM4E
SCHEMBL5205439 0.73 TNFRSF1A (0.51) TUBB4ATUBBTUBA3CTUBA1BTUBA4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1403251-B1 BIS(2-ARYL-5-PYRIDYL) DERIVATIVE KOWA CO (JP) 2007-07-18 EP disclosed
EP-1403251-A1 BIS(2-ARYL-5-PYRIDYL) DERIVATIVE Kowa Co., Ltd. (JP) 2004-03-31 EP disclosed