SCHEMBL5203725

SCHEMBL5203725

CS(=O)(=O)Nc1cc(OCC2=NCCN2)cc(O)c1O

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 11/20 0.49
NISCH Q9Y2I1 7/20 0.48
MAOA P21397 1/20 0.48
MAOB P27338 1/20 0.48
ADRA1D P25100 9/20 0.43
ADRA1B P35368 9/20 0.43
ADRA2A P08913 7/20 0.43
KDM4E B2RXH2 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
TSHR P16473 1/20 0.39
NFKB1 P19838 1/20 0.39
BLM P54132 1/20 0.39
PMP22 Q01453 1/20 0.39
ADRA2C P18825 7/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5201523 0.87 NISCH (0.51) ADRA1ANISCHMAOAMAOBADRA1D
Hydrochloric Acid SCHEMBL5206302 0.86 ADRA1A (0.50) ADRA1ANISCHMAOAMAOBADRA1D
SCHEMBL5200760 0.83 NISCH (0.51) ADRA1ANISCHMAOAMAOBADRA1D
Hydrochloric Acid SCHEMBL5201887 0.82 ADRA1A (0.50) ADRA1ANISCHMAOAMAOBADRA1D
SCHEMBL5206394 0.81 ADRA1A (0.54) ADRA1ANISCHMAOAMAOBADRA1D
Hydrochloric Acid SCHEMBL5201136 0.81 ADRA1A (0.53) ADRA1ANISCHMAOAMAOBADRA1D
SCHEMBL5201006 0.81 ADRA1A (0.62) ADRA1ANISCHMAOAMAOBADRA1D
Hydrochloric Acid SCHEMBL5204266 0.80 ADRA1A (0.61) ADRA1ANISCHMAOAMAOBADRA1D
SCHEMBL5202794 0.78 ADRA1A (0.53) ADRA1ANISCHMAOAMAOBADRA1D
SCHEMBL14340664 0.77 ADRA1A (0.53) ADRA1ANISCHMAOAMAOBADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0887346-B1 N-Phenyl-alkylsulfonamide derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists HOFFMANN LA ROCHE (CH) 2007-12-12 EP disclosed