SCHEMBL5203787

SCHEMBL5203787

CCS(=O)(=O)Nc1cc(CC2=NCCN2)ccc1C

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 9/20 0.49
RAD52 P43351 1/20 0.48
TAAR1 Q96RJ0 4/20 0.47
CYP2D6 P10635 2/20 0.47
NFKB1 P19838 1/20 0.47
HTR1B P28222 7/20 0.45
ADRA2C P18825 4/20 0.45
ADRA2B P18089 3/20 0.45
ADRA2A P08913 3/20 0.45
ADRA1D P25100 3/20 0.45
ADRA1A P35348 3/20 0.45
ADRA1B P35368 3/20 0.45
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5200888 0.89 RAD52 (0.49) HTR1DRAD52TAAR1CYP2D6NFKB1
Hydrochloric Acid SCHEMBL5201249 0.88 RAD52 (0.48) HTR1DRAD52TAAR1CYP2D6NFKB1
SCHEMBL14092040 0.84 RAD52 (0.50) HTR1DRAD52TAAR1CYP2D6NFKB1
SCHEMBL14092056 0.82 LMNA (0.52) HTR1DRAD52TAAR1CYP2D6NFKB1
SCHEMBL4993472 0.79 RAD52 (0.49) HTR1DRAD52TAAR1CYP2D6NFKB1
SCHEMBL11442256 0.77 TAAR1 (0.60) HTR1DTAAR1CYP2D6NFKB1HTR1B
Hydrochloric Acid SCHEMBL11259025 0.76 TAAR1 (0.59) HTR1DTAAR1CYP2D6NFKB1HTR1B
SCHEMBL5203427 0.76 RAD52 (0.48) HTR1DRAD52TAAR1CYP2D6NFKB1
SCHEMBL5203954 0.76 ADRA1A (0.51) HTR1DRAD52TAAR1CYP2D6NFKB1
SCHEMBL5203274 0.76 ADRA1A (0.55) HTR1DRAD52TAAR1CYP2D6NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0887346-B1 N-Phenyl-alkylsulfonamide derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists HOFFMANN LA ROCHE (CH) 2007-12-12 EP disclosed