SCHEMBL5205294

SCHEMBL5205294

Cc1ccc(Oc2cnc(N)nc2NCCO)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 1/20 0.40
MAPT P10636 4/20 0.40
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 2/20 0.39
HSD17B10 Q99714 2/20 0.39
NUDT1 P36639 2/20 0.39
KCNH2 Q12809 2/20 0.38
SCN5A Q14524 2/20 0.38
SCN9A Q15858 2/20 0.38
MEN1 O00255 2/20 0.37
TSHR P16473 2/20 0.37
KMT2A Q03164 2/20 0.37
USP2 O75604 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
CASP1 P29466 1/20 0.37
CASP7 P55210 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TNF P01375 1/20 0.37
PGK1 P00558 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1375252 0.88 MAPT (0.41) MAPTALDH1A1MEN1TSHRKMT2A
SCHEMBL5205013 0.87 KCNH2 (0.40) MAPTALDH1A1KDM4EKCNH2SCN5A
SCHEMBL5206828 0.87 MAPT (0.39) MAPTALDH1A1KDM4EMEN1TSHR
SCHEMBL1376217 0.80 NUDT1 (0.43) MAPTNUDT1KCNH2SCN5ASCN9A
SCHEMBL23472667 0.79 TNF (0.49) NUDT1TSHRUSP2TNF
SCHEMBL5202871 0.79 STK17A (0.42) MAPTNUDT1KCNH2SCN5ASCN9A
SCHEMBL5204559 0.78 STK17A (0.41) MAPTNUDT1KCNH2SCN5ASCN9A
SCHEMBL1376082 0.78 STK17A (0.41) MAPTNUDT1KCNH2SCN5ASCN9A
SCHEMBL1376097 0.78 STK17A (0.41) MAPTNUDT1KCNH2SCN5ASCN9A
SCHEMBL5207953 0.77 SLC6A2 (0.44) ALDH1A1NUDT1KCNH2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165523-B1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC (US) 2007-11-07 EP claimed
EP-1165523-B1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC (US) 2007-11-07 EP disclosed
US-6916820-B1 Neurotrophic substituted pyrimidines KRENITSKY PHARMACEUTICALS, INC. (US) 2005-07-12 US disclosed