SCHEMBL5207953

SCHEMBL5207953

Cc1cc(Cl)ccc1Oc1cnc(N)nc1NCCO

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 8/20 0.44
SLC6A4 P31645 8/20 0.44
SLC6A3 Q01959 6/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
KCNH2 Q12809 2/20 0.39
POLB P06746 1/20 0.39
ALDH1A1 P00352 1/20 0.38
ICAM1 P05362 1/20 0.38
SELE P16581 1/20 0.38
NUDT1 P36639 1/20 0.38
IRAK4 Q9NWZ3 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5203455 0.88 TTR (0.40) SLC6A2SLC6A4SLC6A3CYP2C19L3MBTL1
SCHEMBL5207181 0.86 BCL6 (0.40) SLC6A2SLC6A4SLC6A3CYP2C19KCNH2
SCHEMBL5205013 0.82 KCNH2 (0.40) CYP1A2CYP2C19KCNH2POLBALDH1A1
SCHEMBL5206090 0.80 BCL6 (0.42) SLC6A2SLC6A4SLC6A3CYP2C19ALDH1A1
SCHEMBL6474741 0.79 SCN5A (0.42) SLC6A2SLC6A4SLC6A3CYP1A2CYP3A4
SCHEMBL7510625 0.77 RXFP1 (0.41) CYP2C19L3MBTL1ALDH1A1NUDT1
SCHEMBL5205294 0.77 MMP13 (0.40) KCNH2ALDH1A1NUDT1NPSR1
SCHEMBL6474559 0.77 GAA (0.43) SLC6A2SLC6A4SLC6A3CYP1A2CYP3A4
SCHEMBL5206507 0.76 SLC6A2 (0.39) SLC6A2SLC6A4SLC6A3CYP1A2CYP3A4
SCHEMBL1376410 0.76 MERTK (0.39) SLC6A2SLC6A4SLC6A3CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165523-B1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC (US) 2007-11-07 EP claimed
EP-1165523-B1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC (US) 2007-11-07 EP disclosed
US-6916820-B1 Neurotrophic substituted pyrimidines KRENITSKY PHARMACEUTICALS, INC. (US) 2005-07-12 US disclosed