SCHEMBL5205525

SCHEMBL5205525

Cc1ccc(-c2ccc3c(c2)C=C(C(=O)O)CCN3C)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.39
NOTUM Q6P988 1/20 0.37
KDM4E B2RXH2 2/20 0.36
HDAC4 P56524 1/20 0.34
DHODH Q02127 1/20 0.34
CCR5 P51681 4/20 0.34
CHRNA7 P36544 1/20 0.34
BRD4 O60885 1/20 0.34
BRD2 P25440 1/20 0.34
BRD3 Q15059 1/20 0.34
AKR1C2 P52895 1/20 0.33
AKR1C1 Q04828 1/20 0.33
SRD5A1 P18405 1/20 0.33
ALDH1A1 P00352 2/20 0.33
TSHR P16473 2/20 0.33
NPC1 O15118 1/20 0.33
TP53 P04637 1/20 0.33
HPGD P15428 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27520896 0.85 KDM4E (0.39) KDM4EHDAC4CCR5ALDH1A1TP53
SCHEMBL5206950 0.83 SRD5A1 (0.38) NOTUMKDM4ECCR5SRD5A1ALDH1A1
SCHEMBL5240544 0.80 MYC (0.39) MCL1KDM4ESRD5A1ALDH1A1HPGD
SCHEMBL3498780 0.79 MAPT (0.34) MCL1KDM4ECYP11B1CYP11B2
Hydrochloric Acid SCHEMBL5204621 0.78 MYC (0.38) MCL1SRD5A1ALDH1A1HPGDSMN1; SMN2
SCHEMBL3499816 0.74 CCR5 (0.53) MCL1CCR5ALDH1A1NPC1RAB9A
SCHEMBL6350453 0.73 MAPT (0.41) MCL1TP53RAB9ASMN1; SMN2CYP11B1
SCHEMBL5549419 0.72 TNKS (0.41) MCL1KDM4ESRD5A1ALDH1A1TSHR
SCHEMBL5549424 0.72 TNKS (0.41) MCL1KDM4ESRD5A1ALDH1A1TSHR
SCHEMBL3499129 0.72 MCL1 (0.40) MCL1DHODHCCR5AKR1C2AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040103-B1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2007-03-14 EP disclosed
US-6413947-B1 Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-02 US disclosed