SCHEMBL5206950

SCHEMBL5206950

Cc1ccc(-c2ccc3c(c2)C=C(C(=O)OC(C)(C)C)CCN3C)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 1/20 0.38
GABRA1 P14867 3/20 0.33
GABRG2 P18507 3/20 0.33
GABRB3 P28472 3/20 0.33
GABRA5 P31644 3/20 0.33
GABRA3 P34903 3/20 0.33
WDR5 P61964 1/20 0.33
GABRA2 P47869 1/20 0.33
GABRA4 P48169 1/20 0.33
ALDH1A1 P00352 2/20 0.33
PTPN2 P17706 1/20 0.33
PTPN1 P18031 1/20 0.33
PTPN6 P29350 1/20 0.33
GPR119 Q8TDV5 1/20 0.33
MAPT P10636 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
HSD17B10 Q99714 1/20 0.33
NOTUM Q6P988 1/20 0.33
MMP13 P45452 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5206037 0.86 GPR119 (0.41) SRD5A1ALDH1A1GPR119MAPTTSHR
SCHEMBL5205525 0.83 MCL1 (0.39) SRD5A1ALDH1A1TSHRNOTUMKDM4E
SCHEMBL5206682 0.82 GABRA1 (0.43) SRD5A1GABRA1GABRG2GABRB3GABRA5
Hydrochloric Acid SCHEMBL3499431 0.82 MCL1 (0.38) SRD5A1ALDH1A1TSHRNOTUMKDM4E
SCHEMBL5210235 0.73 CCR5 (0.48) ALDH1A1CA12CA9CCR5
SCHEMBL8130465 0.70 MEN1 (0.33) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL5240927 0.70 MAPT (0.36) GABRA2ALDH1A1MAPTTSHRKDM4E
SCHEMBL6349341 0.69 CCR5 (0.49) CCR5
SCHEMBL6343215 0.69 GABRA1 (0.38) SRD5A1GABRA1GABRG2GABRB3GABRA5
SCHEMBL1808428 0.69 KDM4E (0.38) SRD5A1ALDH1A1TSHRHSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040103-B1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2007-03-14 EP disclosed
US-6413947-B1 Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-02 US disclosed
US-6268354-B1 Pharmaceutical composition for antagonizing CCR5 comprising anilide derivative TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-07-31 US disclosed
US-6172061-B1 AIDS THERAPY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed
US-6166006-A Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-12-26 US disclosed