SCHEMBL5206178

SCHEMBL5206178

Cc1nc(C(F)(F)F)c(C(N)=O)s1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.55
POLB P06746 1/20 0.55
ALDH1A1 P00352 2/20 0.52
KDM4E B2RXH2 2/20 0.48
HTT P42858 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
GAA P10253 3/20 0.44
HSD11B1 P28845 1/20 0.44
CDK8 P49336 1/20 0.42
CDK19 Q9BWU1 1/20 0.42
COMT P21964 1/20 0.38
P2RY1 P47900 1/20 0.37
LIMK1 P53667 3/20 0.35
IKBKB O14920 2/20 0.35
CHUK O15111 1/20 0.34
PRKACA P17612 1/20 0.34
PRKACG P22612 1/20 0.34
PRKACB P22694 1/20 0.34
BTK Q06187 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL975710 0.83 MAPT (0.60) MAPTPOLBALDH1A1KDM4EHTT
SCHEMBL14269337 0.83 MAPT (0.56) MAPTPOLBALDH1A1KDM4EHTT
SCHEMBL2199155 0.81 MAPT (0.56) MAPTPOLBALDH1A1KDM4EHTT
SCHEMBL16217224 0.80 MAPT (0.54) MAPTPOLBALDH1A1KDM4EHTT
SCHEMBL20782350 0.79 CDK8 (0.37) MAPTPOLBALDH1A1KDM4EHTT
SCHEMBL11330712 0.79 ALDH1A1 (0.41) MAPTPOLBALDH1A1CDK8CDK19
SCHEMBL12883301 0.79 MAPT (0.52) MAPTPOLBALDH1A1KDM4EHTT
SCHEMBL13544346 0.79 MAPT (0.52) MAPTPOLBALDH1A1KDM4EHTT
SCHEMBL7988803 0.79 MAPT (0.52) MAPTPOLBALDH1A1KDM4EHTT
SCHEMBL8551963 0.78 MEN1 (0.48) MAPTPOLBALDH1A1KDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108440444-B 2-methyl-4-trifluoromethyl-5-thiazole formamide compound 江苏再拓生物科技有限公司 2021-01-19 CN claimed
CN-111233787-A Green pesticide composition and preparation method thereof 湖南博隽生物医药有限公司 2020-06-05 CN claimed
CN-111226949-A Environment-friendly plant bactericide 湖南博隽生物医药有限公司 2020-06-05 CN claimed
CN-108440444-A 2-methyl-4-trifluoromethyl-5-thiazole formamide compound 湖南博隽生物医药有限公司 2018-08-24 CN claimed
US-9382197-B2 Substituted hydroxamic acids and uses thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2016-07-05 US claimed
CN-1069902-C Thifluzamide with stabilized efficacy ROHM & HAAS (US) 2001-08-22 CN claimed
CN-118420560-A Synthesis method of 2- (trifluoromethyl) -4, 5-disubstituted thiazole compound 西北师范大学 2024-08-02 CN disclosed
CN-112204009-B Modulators of integrated stress pathways 卡里科生命科学有限责任公司 2024-05-07 CN disclosed
CN-117551037-A Compounds as succinate dehydrogenase inhibitors and uses thereof 华东理工大学 2024-02-13 CN disclosed
CN-109641854-B Modulators of integrated stress pathways 卡里科生命科学有限责任公司 2023-02-03 CN disclosed
CN-109195965-B Inhibitors of WDR5 protein-protein binding 普罗佩纶治疗公司 2022-07-26 CN disclosed
CN-108440444-B 2-methyl-4-trifluoromethyl-5-thiazole formamide compound 江苏再拓生物科技有限公司 2021-01-19 CN disclosed
CN-111226949-A Environment-friendly plant bactericide 湖南博隽生物医药有限公司 2020-06-05 CN disclosed
US-20050215495-A1 Macrolide antibiotics ALIHODZIC SULEJMAN 2005-09-29 US disclosed
US-20040077557-A1 Macrolide antibiotics GLAXO GROUP LIMITED (GB) 2004-04-22 US disclosed
EP-1363925-A1 MACROLIDE ANTIBIOTICS GLAXO GROUP LIMITED (GB) 2003-11-26 EP disclosed
WO-2002050091-A1 MACROLIDE ANTIBIOTICS GLAXO GROUP LIMITED (GB) 2002-06-27 WO disclosed
CN-1338452-A Substituted phenylamine derivatives MITSUI CHEMICALS INC (JP) 2002-03-06 CN disclosed
CN-1067063-C Substituted carboxanilide derivatives and plant disease control agents containing the same as active ingredient MITSUI TOATSU CHEMICALS (JP) 2001-06-13 CN disclosed
CN-1178791-A Substituted carboxanilide derivatives and plant disease control agents containing the same as active ingredient MITSUI TOATSU CHEMICALS (JP) 1998-04-15 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050215495-A1 Macrolide antibiotics IL1R1, MRPL12, RPS21 MAPT 3557/4885POLB 2625/4885ALDH1A1 2549/4885
US-20040077557-A1 Macrolide antibiotics MALT1, MRPL21, IL1R1 MAPT 3349/4885POLB 2847/4885ALDH1A1 2482/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.