SCHEMBL5206478

SCHEMBL5206478

Cc1ccc(-c2ccc3c(c2)C=C(C(=O)O)C3)cc1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.45
CCR5 P51681 12/20 0.42
DHODH Q02127 1/20 0.38
AKR1C2 P52895 1/20 0.38
AKR1C1 Q04828 1/20 0.38
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
CCR2 P41597 3/20 0.37
CCR7 P32248 2/20 0.37
CXCR3 P49682 2/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ALPL P05186 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5205124 0.86 CCR5 (0.51) MCL1CCR5CCR2CCR7CXCR3
SCHEMBL3499816 0.84 CCR5 (0.53) MCL1CCR5CCR2CCR7CXCR3
SCHEMBL28745964 0.81 TAAR1 (0.41) CCR5
Biphenyl SCHEMBL27655126 0.75 MAOA (0.59) MCL1MAOAMAOBSMN1; SMN2
SCHEMBL19718183 0.75 ALDH1A1 (0.47) ALDH1A1
SCHEMBL3499773 0.75 CCR5 (0.53) MCL1CCR5MAOAMAOBALDH1A1
SCHEMBL3498192 0.75 MCL1 (0.42) MCL1CCR5DHODHAKR1C2AKR1C1
SCHEMBL7931223 0.74 MCL1 (0.41) MCL1CCR5DHODHAKR1C2AKR1C1
SCHEMBL3093660 0.73 SRD5A1 (0.40) MCL1MAOAMAOBALDH1A1SMN1; SMN2
SCHEMBL14310509 0.73 ALDH1A1 (0.42) CCR5AKR1C2RXRARXRBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040103-B1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2007-03-14 EP disclosed
US-6413947-B1 Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-02 US disclosed
US-6268354-B1 Pharmaceutical composition for antagonizing CCR5 comprising anilide derivative TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-07-31 US disclosed
US-6172061-B1 AIDS THERAPY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed
US-6166006-A Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-12-26 US disclosed
EP-1039899-A2 PHARMACEUTICAL COMPOSITION FOR ANTAGONIZING CCR5 COMPRISING ANILIDE DERIVATIVE Takeda Chemical Industries, Ltd. (JP) 2000-10-04 EP disclosed
EP-1040103-A1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-10-04 EP disclosed
WO-1999032100-A2 PHARMACEUTICAL COMPOSITION FOR ANTAGONIZING CCR5 COMPRISING ANILIDE DERIVATIVE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-07-01 WO disclosed
WO-1999032468-A1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-07-01 WO disclosed