SCHEMBL5207314

SCHEMBL5207314

O=C(Nc1ccc2[nH]c(-c3ccccc3)cc2c1)c1ccccc1Cl

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 2/20 0.60
JAK1 P23458 2/20 0.60
NPC1 O15118 2/20 0.60
RAB9A P51151 2/20 0.60
SMO Q99835 7/20 0.57
NR2E3 Q9Y5X4 4/20 0.56
NAMPT P43490 1/20 0.53
KCNK3 O14649 1/20 0.52
KCNK9 Q9NPC2 1/20 0.52
MAPT P10636 2/20 0.51
KDM4E B2RXH2 1/20 0.51
MEN1 O00255 1/20 0.51
ALDH1A1 P00352 1/20 0.51
LMNA P02545 1/20 0.51
CYP19A1 P11511 1/20 0.51
KMT2A Q03164 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
PKM P14618 1/20 0.51
MAOB P27338 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5207022 0.85 MAOA (0.55) NPC1RAB9ANR2E3NAMPTKCNK3
SCHEMBL5208301 0.82 KCNK3 (0.57) NPC1RAB9AKCNK3KCNK9MAPT
SCHEMBL15060321 0.82 NAMPT (0.59) NPC1RAB9ANAMPTMAPTKDM4E
SCHEMBL4464384 0.81 KIT (0.67) JAK2JAK1NPC1RAB9ASMO
SCHEMBL14182736 0.80 MAOA (0.67) JAK2NPC1RAB9ANAMPTMAPT
SCHEMBL14182739 0.79 MAOA (0.59) JAK2NPC1RAB9AMAPTKDM4E
SCHEMBL18145948 0.77 MEN1 (0.43) JAK2JAK1NPC1RAB9ANR2E3
SCHEMBL21022000 0.77 NAMPT (0.42) JAK2JAK1NPC1RAB9ANR2E3
SCHEMBL18145945 0.77 MEN1 (0.43) JAK2JAK1NPC1RAB9ANR2E3
SCHEMBL28671945 0.76 GUSB (0.53) NPC1RAB9ANAMPTMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833829-A2 BENZAMIDE SUBSTITUTED IMIDAZO- AND PYRROLO-PYRIDINES AS PROTEIN KINASE INHIBITORS F. Hoffmann-Roche AG (CH) 2007-09-19 EP disclosed
WO-2006066913-A2 BENZAMIDE SUBSTITUTED IMIDAZO- AND PYROLO-PYRIDINES AS PROTEIN KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2006-06-29 WO disclosed