SCHEMBL5207326

SCHEMBL5207326

CC(C)Cn1c(S(C)(=O)=O)nc(OCc2ccc(F)cc2F)cc1=O

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.38
MAPK14 Q16539 12/20 0.37
IDH1 O75874 1/20 0.35
IDO1 P14902 1/20 0.35
AGXT P21549 1/20 0.35
PTGS2 P35354 1/20 0.35
P2RX3 P56373 1/20 0.35
PTGER1 P34995 1/20 0.35
CYP1A1 P04798 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP1B1 Q16678 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5207452 0.84 MEN1 (0.39) MAOBMAPK14IDH1IDO1AGXT
SCHEMBL5204609 0.80 MCHR1 (0.38) MAOBMAPK14
SCHEMBL5207062 0.78 MAPK14 (0.38) MAPK14
SCHEMBL3523048 0.72 MAPK14 (0.39) MAOBMAPK14PTGER1
SCHEMBL5205590 0.72 MAOB (0.39) MAOBMAPK14IDO1AGXTPTGER1
SCHEMBL5202380 0.72 MAOB (0.42) MAOBMAPK14IDO1AGXTPTGER1
SCHEMBL5203583 0.72 MAPK14 (0.43) MAPK14
SCHEMBL5207124 0.72 MAPK14 (0.43) MAPK14PTGER1
SCHEMBL5203024 0.71 MAOB (0.37) MAOBMAPK14IDO1AGXTPTGER1
SCHEMBL5203740 0.71 CYP1A1 (0.42) MAOBMAPK14PTGER1CYP1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1802590-A1 SUBSTITUTED N-ALKYLPYRIMIDINONES Pharmacia & Upjohn Company LLC (US) 2007-07-04 EP disclosed
WO-2006040666-A1 SUBSTITUTED N-ALKYLPYRIMIDINONES PHARMACIA & UPJOHN COMPANY LLC (US) 2006-04-20 WO disclosed