SCHEMBL5207780

SCHEMBL5207780

COc1cc(Cl)c[c]c1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.37
ERN1 O75460 1/20 0.36
CXCL12 P48061 1/20 0.36
ACHE P22303 2/20 0.34
KDM4E B2RXH2 3/20 0.34
MAPT P10636 3/20 0.34
HSP90AA1 P07900 2/20 0.34
S1PR4 O95977 1/20 0.34
G6PD P11413 1/20 0.34
S1PR1 P21453 1/20 0.34
MAPK1 P28482 1/20 0.34
OPRK1 P41145 1/20 0.34
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.34
CACNA1B Q00975 1/20 0.34
APBA1 Q02410 1/20 0.34
MCL1 Q07820 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
APOBEC3G Q9HC16 1/20 0.34
TLR9 Q9NR96 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2349873 0.79 TRPV4 (0.38) TRPV4ERN1CXCL12ACHEKDM4E
SCHEMBL1491051 0.79 ACHE (0.46) ERN1ACHEMAPTMAPK1NPSR1
SCHEMBL1810937 0.77 CA12 (0.43) ACHEKDM4EMAPTMAPK1GAA
SCHEMBL28805089 0.76 POLB (0.39) ERN1ACHEKDM4EMAPTNPSR1
SCHEMBL1639475 0.76 ERN1 (0.43) TRPV4ERN1CXCL12KDM4EMAPT
SCHEMBL27695180 0.76 TRPV4 (0.36) TRPV4ERN1KDM4EMAPTHSP90AA1
SCHEMBL2344974 0.76 TRPV4 (0.36) TRPV4ERN1KDM4EMAPTHSP90AA1
SCHEMBL27743323 0.71 TAAR1 (0.37) TRPV4ERN1KDM4EMAPTHSP90AA1
SCHEMBL3702697 0.70
SCHEMBL13256218 0.70 ERN1 (0.45) TRPV4ERN1CXCL12ACHEKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0980867-B1 KETONE DERIVATIVES AND MEDICINAL USE THEREOF TORAY INDUSTRIES (JP) 2007-08-08 EP disclosed
US-6184245-B1 Cyclic ketone derivatives and their medical applications TORAY INDUSTRIES INC. (JP) 2001-02-06 US disclosed
US-6100292-A Ketone derivatives and their medical applications TORAY INDUSTRIES, INC. (JP) 2000-08-08 US disclosed
EP-0980867-A1 KETONE DERIVATIVES AND MEDICINAL USE THEREOF TORAY INDUSTRIES, INC. (JP) 2000-02-23 EP disclosed
EP-0962456-A1 CYCLIC KETONE DERIVATIVE AND PHARMACEUTICAL USE THEREOF TORAY INDUSTRIES, INC. (JP) 1999-12-08 EP disclosed