SCHEMBL5207841

SCHEMBL5207841

CS(=O)(=O)c1ccc(Cn2ncnc2-c2ccccc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.58
HDAC6 Q9UBN7 2/20 0.58
PTGS2 P35354 13/20 0.52
PTGS1 P23219 6/20 0.52
PTGDR2 Q9Y5Y4 3/20 0.46
P2RX7 Q99572 1/20 0.45
DHFR P00374 1/20 0.43
GHSR Q92847 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10771603 0.77 PTGDR2 (0.44) PTGS2PTGS1PTGDR2
SCHEMBL31272227 0.75 HDAC1 (0.57) HDAC1HDAC6P2RX7
SCHEMBL7490899 0.73 HDAC1 (0.45) HDAC1HDAC6PTGS2PTGDR2P2RX7
SCHEMBL6601374 0.69 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL6601664 0.69 PTGS2 (0.75) PTGS2PTGS1
SCHEMBL29114966 0.68 PTGS2 (0.60) HDAC6PTGS2PTGS1
SCHEMBL12597163 0.68 NPC1 (0.56) HDAC1HDAC6P2RX7
SCHEMBL3429586 0.68 PTGER4 (0.55) PTGS2PTGS1PTGDR2
SCHEMBL9328526 0.67 HDAC1 (0.55) HDAC1HDAC6PTGS2PTGDR2
SCHEMBL10304515 0.67 HDAC1 (0.48) HDAC1HDAC6P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1458706-B1 DIARYL 1,2,4-TRIAZOLE DERIVATIVES AS A HIGHLY SELECTIVE CYCLOOXYGENASE-2 INHIBITOR CJ CORP (KR) 2007-07-11 EP disclosed