SCHEMBL5209478

SCHEMBL5209478

COC(=O)C1=Cc2cc(-c3ccc4c(c3)OCO4)ccc2OCC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.44
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 3/20 0.44
MAPT P10636 3/20 0.44
MEN1 O00255 2/20 0.44
TP53 P04637 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
GAA P10253 1/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
CASP1 P29466 1/20 0.44
CASP7 P55210 1/20 0.44
HSD17B10 Q99714 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
NPC1 O15118 7/20 0.43
RAB9A P51151 5/20 0.43
CCR5 P51681 6/20 0.43
ADORA3 P0DMS8 2/20 0.43
ADORA1 P30542 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7685102 0.86 CCR5 (0.46) CCR5CA12CA9
SCHEMBL5204016 0.85 ALDH1A1 (0.45) KMT2AKDM4EALDH1A1MAPTMEN1
SCHEMBL5209473 0.83 CCR5 (0.40) CCR5CA12CA9
SCHEMBL5211895 0.82 NR4A2 (0.42) KDM4ECCR5CA12CA9
SCHEMBL5206762 0.81 NPC1 (0.43) KMT2AKDM4EALDH1A1MAPTMEN1
SCHEMBL7975074 0.81 KMT2A (0.41) KMT2AKDM4EALDH1A1MAPTMEN1
SCHEMBL7700889 0.80 CA12 (0.63) KMT2AKDM4EALDH1A1MAPTMEN1
SCHEMBL5209506 0.80 CCR2 (0.46) MAPTTP53CA12CA9
SCHEMBL5209410 0.79 CA12 (0.41) CCR5CA12CA9
SCHEMBL7674673 0.78 CA12 (0.43) CCR5CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040103-B1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2007-03-14 EP disclosed
US-6413947-B1 Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-02 US disclosed
US-6268354-B1 Pharmaceutical composition for antagonizing CCR5 comprising anilide derivative TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-07-31 US disclosed
US-6172061-B1 AIDS THERAPY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed
US-6166006-A Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-12-26 US disclosed