SCHEMBL5210693

SCHEMBL5210693

COC(=O)CCc1oc(-n2ccnc2CO)nc1-c1ccc(Cl)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
KDM4E B2RXH2 4/20 0.40
MAPT P10636 3/20 0.40
LMNA P02545 2/20 0.40
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
HSP90AA1 P07900 1/20 0.33
HSP90B1 P14625 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
GAA P10253 2/20 0.33
HPGD P15428 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
EGFR P00533 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6603683 0.88 ALDH1A1 (0.39) ALDH1A1KDM4EMAPTLMNACYP11B1
SCHEMBL5208221 0.88 RXRA (0.43) ALDH1A1KDM4EMAPTLMNAHPGD
SCHEMBL5206976 0.86 KMT2A (0.38) ALDH1A1KDM4EMAPTLMNACYP11B1
SCHEMBL5211827 0.85 ALDH1A1 (0.37) ALDH1A1KDM4EMAPTLMNACYP11B1
SCHEMBL1360319 0.82 TP53 (0.38) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL7453572 0.81 RXRA (0.43) ALDH1A1KDM4EMAPTHPGDRXRA
SCHEMBL7462798 0.80 RXRA (0.42) ALDH1A1KDM4EMAPTHPGDRXRA
SCHEMBL5211741 0.80 POLB (0.38) MAPTLMNAMEN1KMT2AGAA
SCHEMBL5211444 0.79 CYP11B1 (0.42) ALDH1A1KDM4EMAPTLMNACYP11B1
SCHEMBL1360271 0.78 RXRA (0.38) MAPTMEN1KMT2AHPGDCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7183276-B2 Azole compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-27 US disclosed
US-20050090534-A1 Azole compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-04-28 US disclosed
EP-1486490-A1 AZOLE COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2004-12-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050090534-A1 Azole compounds AHR, NR0B2, NR2C2 ALDH1A1 1651/4885KDM4E 2428/4885MAPT 3958/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.