SCHEMBL5211007

SCHEMBL5211007

C[C@H]1Oc2ccc(CNCCCC(F)(F)F)cc2N=C1N

nearest known ligand 0.36

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 5/20 0.36
NOS1 P29475 5/20 0.36
NOS2 P35228 5/20 0.36
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5241724 1.00 NOS3 (0.36) NOS3NOS1NOS2PARP1
Hydrochloric Acid SCHEMBL5189277 0.99 NOS3 (0.37) NOS3NOS1NOS2PARP1
Hydrochloric Acid SCHEMBL5188387 0.99 NOS3 (0.37) NOS3NOS1NOS2PARP1
Hydrochloric Acid SCHEMBL5189228 0.89 NOS1 (0.33) NOS3NOS1NOS2
SCHEMBL7843673 0.86 MC4R (0.43) NOS3NOS1NOS2PARP1
Hydrochloric Acid SCHEMBL6308988 0.85 MC4R (0.42) NOS3NOS1NOS2PARP1
Hydrochloric Acid SCHEMBL5189703 0.85 BACE1 (0.38) NOS3NOS1NOS2PARP1
Hydrochloric Acid SCHEMBL5470037 0.85 NOS3 (0.35) NOS3NOS1NOS2PARP1
Hydrochloric Acid SCHEMBL6305979 0.84 NOS3 (0.38) NOS3NOS1NOS2PARP1
Hydrochloric Acid SCHEMBL5189769 0.84 NOS1 (0.36) NOS3NOS1NOS2PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1282610-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THE USE THEREOF IN MEDICAMENTS BAYER SCHERING PHARMA AG (DE) 2007-07-25 EP claimed