SCHEMBL7843673

SCHEMBL7843673

CC1Oc2ccc(CNCCCN)cc2N=C1N

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MC4R P32245 2/20 0.43
MC5R P33032 2/20 0.43
MC3R P41968 1/20 0.43
NOS1 P29475 6/20 0.38
NOS3 P29474 5/20 0.38
NOS2 P35228 5/20 0.38
PARP1 P09874 1/20 0.36
KAT2B Q92831 1/20 0.33
CXCR4 P61073 1/20 0.32
MAOB P27338 1/20 0.32
KDM4E B2RXH2 1/20 0.31
POLB P06746 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
EP300 Q09472 1/20 0.31
CHRM2 P08172 1/20 0.31
ROCK2 O75116 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6308988 0.99 MC4R (0.42) MC4RMC5RMC3RNOS1NOS3
Hydrochloric Acid SCHEMBL6608313 0.93 MC4R (0.38) MC4RMC5RMC3RNOS1NOS3
Hydrochloric Acid SCHEMBL6305979 0.88 NOS3 (0.38) MC4RMC5RMC3RNOS1NOS3
Hydrochloric Acid SCHEMBL5189769 0.88 NOS1 (0.36) MC4RMC5RNOS1NOS3NOS2
SCHEMBL6611984 0.87 PARP1 (0.45) NOS1NOS3NOS2PARP1KDM4E
SCHEMBL5241724 0.86 NOS3 (0.36) NOS1NOS3NOS2PARP1
SCHEMBL5211007 0.86 NOS3 (0.36) NOS1NOS3NOS2PARP1
Hydrochloric Acid SCHEMBL6302797 0.86 PARP1 (0.44) NOS1NOS3NOS2PARP1ROCK2
Hydrochloric Acid SCHEMBL5189277 0.85 NOS3 (0.37) NOS1NOS3NOS2PARP1CYP1A2
Hydrochloric Acid SCHEMBL5188387 0.85 NOS3 (0.37) NOS1NOS3NOS2PARP1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1319097-A Benzoxazine and benzothiazine derivatives and their use in medicines SCHERING AG (DE) 2001-10-24 CN disclosed
EP-1114037-A1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN MEDICINES Schering Aktiengesellschaft (DE) 2001-07-11 EP disclosed
WO-2000017173-A1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN MEDICINES SCHERING AKTIENGESELLSCHAFT (DE) 2000-03-30 WO disclosed