SCHEMBL5212357

SCHEMBL5212357

CC(C)CN1C(C(=O)O)CC(c2cnccn2)C1c1csc(-c2ccccc2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CPT1A P50416 4/20 0.38
CPT1B Q92523 3/20 0.38
CPT2 P23786 2/20 0.37
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
CYP19A1 P11511 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HTT P42858 1/20 0.35
CTSK P43235 1/20 0.35
CCR5 P51681 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
TP53 P04637 1/20 0.33
TACR3 P29371 1/20 0.33
DPP4 P27487 1/20 0.33
DPP8 Q6V1X1 1/20 0.33
DPP9 Q86TI2 1/20 0.33
KCNJ6 P48051 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5212350 1.00 CPT1A (0.38) CPT1ACPT1BCPT2NPC1RAB9A
SCHEMBL6636875 0.72 CYP19A1 (0.42) CPT1ACPT1BCPT2NPC1RAB9A
SCHEMBL5641473 0.71 SMN1; SMN2 (0.36) CPT1ACPT1BCPT2NPC1RAB9A
SCHEMBL14443179 0.69 CPT1A (0.36) CPT1ACPT1BCPT2NPC1RAB9A
SCHEMBL5219538 0.69 ABL1 (0.34) CPT1ACPT1BCPT2NPC1RAB9A
SCHEMBL13643056 0.59 KDM4E (0.55) NPC1RAB9ASMN1; SMN2MAPTKDM4E
SCHEMBL1667203 0.58 KDM4E (0.41) KDM4E
SCHEMBL1667202 0.58 KDM4E (0.41) KDM4E
SCHEMBL31076264 0.58 KDM4E (0.41) KDM4E
SCHEMBL4713366 0.57 CTSK (0.70) NPC1RAB9ASMN1; SMN2MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1440069-B1 4-(6-MEMBERED)-HETEROARYL ACYL PYRROLIDINE DERIVATIVES AS HCV INHIBITORS GLAXO GROUP LTD (GB) 2007-08-15 EP disclosed