SCHEMBL6636875

SCHEMBL6636875

O=C(O)C1CC(c2cnccn2)C(c2csc(-c3ccccc3)n2)N1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 5/20 0.42
RAB9A P51151 3/20 0.42
NPC1 O15118 2/20 0.42
CPT1A P50416 3/20 0.40
CPT1B Q92523 2/20 0.40
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 1/20 0.39
AXL P30530 1/20 0.38
PBRM1 Q86U86 1/20 0.38
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
HPGDS O60760 1/20 0.38
IRAK4 Q9NWZ3 1/20 0.38
TLR7 Q9NYK1 2/20 0.37
CPT2 P23786 1/20 0.37
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
LMNA P02545 1/20 0.36
AR P10275 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6633356 0.81 KDM4E (0.37) RAB9AKDM4EALDH1A1MAPTLMNA
SCHEMBL6632885 0.76 HTT (0.41) RAB9ANPC1KDM4EALDH1A1TP53
SCHEMBL5196351 0.75 ALDH1A1 (0.33) RAB9AKDM4EALDH1A1MAPTLMNA
SCHEMBL5641473 0.73 SMN1; SMN2 (0.36) CYP19A1RAB9ANPC1CPT1ACPT1B
SCHEMBL5212357 0.72 CPT1A (0.38) CYP19A1RAB9ANPC1CPT1ACPT1B
SCHEMBL5212350 0.72 CPT1A (0.38) CYP19A1RAB9ANPC1CPT1ACPT1B
SCHEMBL6633848 0.71 KDM4E (0.32) KDM4EALDH1A1
SCHEMBL14443179 0.69 CPT1A (0.36) CYP19A1RAB9ANPC1CPT1ACPT1B
SCHEMBL21409140 0.62 CYP1A2 (0.40) KDM4EALDH1A1MAPTLMNA
SCHEMBL21409139 0.62 CYP1A2 (0.40) KDM4EALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1440069-A1 4-(6-MEMBERED)-HETEROARYL ACYL PYRROLIDINE DERIVATIVES AS HCV INHIBITORS GLAXO GROUP LIMITED (GB) 2004-07-28 EP disclosed
WO-2003037895-A1 4-(6-MEMBERED)-HETEROARYL ACYL PYRROLIDINE DERIVATIVES AS HCV INHIBITORS GLAXO GROUP LIMITED (GB) 2003-05-08 WO disclosed