SCHEMBL5215870

SCHEMBL5215870

C1=CC2(c3ccc(-c4csc5ccccc45)nc3)CCN(C1)C2

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.44
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
C5AR1 P21730 2/20 0.35
CHRM2 P08172 2/20 0.33
CHRM4 P08173 2/20 0.33
CHRM5 P08912 2/20 0.33
CHRM1 P11229 2/20 0.33
CHRM3 P20309 2/20 0.33
APP P05067 1/20 0.33
CYP2C9 P11712 1/20 0.33
CCNC P24863 1/20 0.32
CDK8 P49336 1/20 0.32
ACVRL1 P37023 1/20 0.32
ACVR1 Q04771 1/20 0.32
ALDH1A1 P00352 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL4474316 0.99 KDM1A (0.43) KDM1ACYP11B1CYP11B2C5AR1CHRM2
SCHEMBL4465415 0.81 NPC1 (0.36) CYP11B1CYP11B2
SCHEMBL4467650 0.81
SCHEMBL4463819 0.79 HSD11B1 (0.38) CYP11B1CYP11B2
SCHEMBL4473740 0.79 KDM1A (0.46) KDM1ACYP11B1CYP11B2C5AR1CHRM2
Bromide SCHEMBL4466117 0.78 HSD11B1 (0.37) CYP11B1CYP11B2
SCHEMBL4467652 0.78 KDM1A (0.43) KDM1ACYP11B1CYP11B2CHRM2CHRM4
SCHEMBL5219426 0.78 HSD11B1 (0.32)
SCHEMBL5217300 0.78 HPGDS (0.37) CYP11B1CYP11B2ALDH1A1HSD17B10
Bromide SCHEMBL4460345 0.77 HSD11B1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465893-B1 DERIVATIVES OF 5-(PYRIDIN-3-YL)-1-AZABICYCLO (3.2.1) OCTANE, THE PREPARATION THEREOF AND THE APPLICATION OF SAME IN THERAPEUTICS SANOFI AVENTIS (FR) 2007-02-28 EP claimed