SCHEMBL5217465

SCHEMBL5217465

C[C@]1(C(=O)OCc2ccccc2)CCCNC1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 1/20 0.47
CRBN Q96SW2 1/20 0.47
ALDH1A1 P00352 1/20 0.44
HTR2C P28335 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5215704 1.00 DDB1 (0.47) DDB1CRBNALDH1A1HTR2C
SCHEMBL5215715 1.00 DDB1 (0.47) DDB1CRBNALDH1A1HTR2C
SCHEMBL23582686 0.92 DDB1 (0.49) DDB1CRBNALDH1A1HTR2C
SCHEMBL12621202 0.84 ALDH1A1 (0.53) DDB1CRBNALDH1A1
SCHEMBL18692576 0.84 ALDH1A1 (0.53) DDB1CRBNALDH1A1
SCHEMBL5213485 0.83 DDB1 (0.51) DDB1CRBNALDH1A1HTR2C
SCHEMBL20221555 0.83 ALDH1A1 (0.51) DDB1CRBNALDH1A1
SCHEMBL8143637 0.81 DDB1 (0.47) DDB1CRBNALDH1A1HTR2C
SCHEMBL8751651 0.81 OPRM1 (0.49) DDB1CRBNALDH1A1
SCHEMBL14650073 0.78 CTSS (0.48) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1322596-B1 ZWITTERIONIC TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2007-08-15 EP disclosed
EP-1322596-A1 ZWITTERIONIC TACHYKININ RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2003-07-02 EP disclosed
US-6479518-B2 PSYCHOLOGICAL DISORDERS MERCK & CO., INC. 2002-11-12 US disclosed
US-20020042431-A1 Zwitterionic tachykinin receptor antagonists MERCK & CO., INC. 2002-04-11 US disclosed
WO-2002024629-A1 ZWITTERIONIC TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2002-03-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020042431-A1 Zwitterionic tachykinin receptor antagonists NPY5R, NPY1R, NPY2R DDB1 4170/4885CRBN 3505/4885ALDH1A1 3769/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.