SCHEMBL5217883

SCHEMBL5217883

CNc1ncc(-c2ccccc2)c(-c2ccccc2)n1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 1/20 0.53
RPS6KA3 P51812 1/20 0.52
ADORA1 P30542 15/20 0.51
ADORA2A P29274 3/20 0.51
PTGS2 P35354 2/20 0.47
TDP1 Q9NUW8 1/20 0.46
ADORA2B P29275 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5214862 0.84 RPS6KA3 (0.70) RPS6KA3ADORA1ADORA2APTGS2ADORA2B
SCHEMBL28360587 0.82 GAA (0.56) ADORA1ADORA2A
SCHEMBL31061144 0.79 ADORA1 (0.55) ADORA1ADORA2APTGS2ADORA2B
SCHEMBL6133449 0.79 ADORA1 (0.41) NUDT1RPS6KA3ADORA1ADORA2ATDP1
SCHEMBL1350076 0.78 AKT1 (0.45) RPS6KA3ADORA1ADORA2A
SCHEMBL6133483 0.78 CYP1A2 (0.50) NUDT1RPS6KA3ADORA1ADORA2APTGS2
SCHEMBL24309336 0.77 ADORA1 (0.46) ADORA1ADORA2APTGS2ADORA2B
SCHEMBL18496447 0.77 ACHE (0.53) RPS6KA3ADORA1ADORA2APTGS2TDP1
SCHEMBL5451373 0.76 ADORA1 (0.53) RPS6KA3ADORA1ADORA2APTGS2ADORA2B
SCHEMBL5451875 0.76 ADORA1 (0.57) ADORA1ADORA2APTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7205302-B2 Anticoagulants; antilipemic agents; cardiovascular disorders NIPPON SHINYAKU CO., LTD. (JP) 2007-04-17 US disclosed
EP-1400518-B1 HETEROCYCLIC COMPOUND DERIVATIVES AND MEDICINES NIPPON SHINYAKU CO LTD (JP) 2007-01-17 EP disclosed
US-20040102436-A1 Heterocyclic compound derivatives and medicines NIPPON SHINYAKU CO., LTD. (JP) 2004-05-27 US disclosed
EP-1400518-A1 HETEROCYCLIC COMPOUND DERIVATIVES AND MEDICINES Nippon Shinyaku Co., Ltd. (JP) 2004-03-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040102436-A1 Heterocyclic compound derivatives and medicines CNR2, CNR1, GPR55 NUDT1 2498/4885RPS6KA3 1852/4885ADORA1 181/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.