SCHEMBL5217971

SCHEMBL5217971

O=CC(Cl)c1cc(Cl)ccc1O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.50
MEN1 O00255 8/20 0.45
KMT2A Q03164 8/20 0.45
HTT P42858 4/20 0.45
MAPT P10636 4/20 0.45
MAPK1 P28482 3/20 0.45
NPSR1 Q6W5P4 2/20 0.45
HSD17B10 Q99714 4/20 0.43
TSHR P16473 3/20 0.43
HPGD P15428 7/20 0.41
ALDH1A1 P00352 6/20 0.41
TDP1 Q9NUW8 4/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
ALOX15 P16050 4/20 0.41
ALOX12 P18054 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
CYP3A4 P08684 4/20 0.39
LMNA P02545 3/20 0.39
HSP90AA1 P07900 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7519487 0.79 KMT2A (0.51) ERN1MEN1KMT2AHTTMAPT
SCHEMBL6819000 0.79 CA3 (0.38) ERN1MEN1KMT2AHSD17B10HPGD
SCHEMBL16881123 0.77 TSHR (0.45) ERN1KMT2AHTTMAPK1HSD17B10
SCHEMBL3978958 0.76 TP53 (0.48) MEN1KMT2AHTTMAPTNPSR1
SCHEMBL19954062 0.75 MEN1 (0.50) ERN1MEN1KMT2AHTTMAPT
SCHEMBL27601029 0.75 ERN1 (0.44) ERN1MEN1KMT2AHTTMAPT
SCHEMBL8813338 0.74 ERN1 (0.43) ERN1MEN1KMT2AHTTMAPT
SCHEMBL26999265 0.74 MAPT (0.48) ERN1MEN1KMT2AHTTMAPT
SCHEMBL25241487 0.74 GABRA1 (0.46) ERN1MEN1KMT2AMAPTHSD17B10
SCHEMBL16093965 0.73 TSHR (0.45) ERN1MEN1KMT2AHTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765810-A1 2,4-DIAMINOQUINAZOLINES FOR SPINAL MUSCULAR ATROPHY Decode Chemistry, Inc. (US) 2007-03-28 EP disclosed
WO-2005123724-A1 2,4-DIAMINOQUINAZOLINES FOR SPINAL MUSCULAR ATROPHY DECODE CHEMISTRY, INC. (US) 2005-12-29 WO disclosed