SCHEMBL5218113

SCHEMBL5218113

Cc1noc(-c2ccc(-c3cc(N)ccc3C)cc2)n1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.71
PIK3CG P48736 8/20 0.47
PIK3CD O00329 7/20 0.47
MTOR P42345 4/20 0.47
MAPT P10636 2/20 0.45
TP53 P04637 1/20 0.45
MAPK14 Q16539 1/20 0.45
LMNA P02545 1/20 0.44
THRB P10828 1/20 0.44
BCHE P06276 2/20 0.44
HTR1A P08908 1/20 0.42
HTR2C P28335 1/20 0.42
NPC1 O15118 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
RAB9A P51151 2/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31415554 0.87 ACHE (0.59) ACHEPIK3CGPIK3CDMTORMAPT
SCHEMBL981283 0.84 ACHE (1.00) ACHEMAPTTP53LMNATHRB
SCHEMBL13415305 0.78 ACHE (0.80) ACHEMAPTTP53LMNATHRB
SCHEMBL21939240 0.78 ACHE (0.59) ACHEPIK3CGPIK3CDMTORMAPT
SCHEMBL27436286 0.78 ACHE (0.64) ACHEPIK3CGPIK3CDMTORMAPT
SCHEMBL30955218 0.78 ACHE (0.64) ACHEPIK3CGPIK3CDMTORMAPT
SCHEMBL5122825 0.77 NR1H4 (0.60) ACHEMAPTTP53MAPK14
SCHEMBL3783964 0.76 ALDH1A1 (0.54) ACHEMAPTTP53LMNANPC1
SCHEMBL2092192 0.75 NPC1 (0.63) ACHEMAPTTP53MAPK14LMNA
SCHEMBL61991 0.74 ACHE (0.64) ACHEMAPTTP53BCHEHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1499600-B1 HETEROARYL SUBSTITUTED BIPHENYL DERIVATIVES AS P38 KINASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2007-07-25 EP disclosed