SCHEMBL5218374

SCHEMBL5218374

Cc1cc(COc2cc(C(=O)O)cc3occc23)no1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 1/20 0.45
HTT P42858 2/20 0.42
ATR Q13535 1/20 0.40
ATRIP Q8WXE1 1/20 0.40
NOX1 Q9Y5S8 1/20 0.40
NOS1 P29475 1/20 0.38
KCNA3 P22001 1/20 0.38
ACACB O00763 2/20 0.37
PPARG P37231 1/20 0.36
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPK1 P28482 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CG P48736 1/20 0.36
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36
MRGPRX4 Q96LA9 2/20 0.35
PKM P14618 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226263 0.89 NOX1 (0.42) PTGER1HTTATRATRIPNOX1
SCHEMBL2654597 0.86 GCK (0.44) HTTNOX1ALDH1A1MAPK1SMN1; SMN2
SCHEMBL5218574 0.84 PTGER1 (0.44) PTGER1HTTATRATRIPNOX1
SCHEMBL2666934 0.81 NOX1 (0.44) HTTNOX1ALDH1A1MAPK1PKM
SCHEMBL5221627 0.79 NOX1 (0.45) HTTNOX1ALDH1A1MAPK1PKM
SCHEMBL14381218 0.78 NOX1 (0.34) PTGER1ATRATRIPNOX1NOS1
SCHEMBL3371103 0.77 HTT (0.60) PTGER1HTTNOX1ALDH1A1MAPK1
SCHEMBL16471641 0.74 KCNA3 (0.44) KCNA3ALDH1A1MAPK1MRGPRX4
SCHEMBL15417869 0.73 REN (0.47) KCNA3PKM
SCHEMBL18585491 0.73 CA12 (0.51) HTTKCNA3ALDH1A1MAPK1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1578745-B1 BENZOFURAN DERIVATivES, PROCESS FOR THEIR PREPARATION AND INTERMEDIATES THEREOF ASTRAZENECA AB (SE) 2007-11-14 EP disclosed