SCHEMBL5219084

SCHEMBL5219084

C/C=C/c1cc(C(=O)OC)c(F)c(N2CCCCS2(=O)=O)c1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSD P07339 3/20 0.36
BACE1 P56817 3/20 0.36
BACE2 Q9Y5Z0 3/20 0.36
PIK3C3 Q8NEB9 1/20 0.34
POLB P06746 2/20 0.34
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
PTGS2 P35354 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
TP53 P04637 2/20 0.33
LDHA P00338 1/20 0.33
CALCA P06881 2/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224665 0.97 PIK3C3 (0.37) CTSDBACE1BACE2PIK3C3KDM4E
SCHEMBL5224667 0.97 PIK3C3 (0.37) CTSDBACE1BACE2PIK3C3KDM4E
SCHEMBL5219078 0.89 PTGS2 (0.33) KDM4ENPC1RAB9ASMN1; SMN2NPSR1
SCHEMBL5219097 0.89 PTGS2 (0.33) KDM4ENPC1RAB9ASMN1; SMN2NPSR1
SCHEMBL5219089 0.89 PTGS2 (0.33) KDM4ENPC1RAB9ASMN1; SMN2NPSR1
SCHEMBL5224678 0.85 PTGS2 (0.34) KDM4ENPC1RAB9ASMN1; SMN2NPSR1
SCHEMBL5224671 0.85 PTGS2 (0.34) KDM4ENPC1RAB9ASMN1; SMN2NPSR1
SCHEMBL5217755 0.83 CTSD (0.37) CTSDBACE1BACE2PIK3C3POLB
SCHEMBL5223229 0.83 KDM4E (0.41) CTSDBACE1BACE2PIK3C3POLB
SCHEMBL5221784 0.80 CTSD (0.42) CTSDBACE1BACE2PIK3C3POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed