SCHEMBL5219882

SCHEMBL5219882

N#Cc1c(F)cccc1OCCc1cccc2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
KDM4E B2RXH2 2/20 0.46
MAPT P10636 2/20 0.44
LMNA P02545 1/20 0.44
TSHR P16473 1/20 0.44
HTT P42858 1/20 0.44
MAOB P27338 1/20 0.43
HTR1B P28222 4/20 0.43
HPGD P15428 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CASP1 P29466 1/20 0.39
S1PR5 Q9H228 4/20 0.39
KCNA3 P22001 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HTR1D P28221 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5217402 0.88 LMNA (0.43) ALDH1A1MAPTLMNATSHRHTT
SCHEMBL5223526 0.83 HSD11B1 (0.43) MAPTLMNATSHRHTTHPGD
SCHEMBL1154474 0.79 CYP11B1 (0.43) ALDH1A1MAPTLMNATSHRHTT
SCHEMBL5216704 0.79 MAPT (0.42) ALDH1A1KDM4EMAPTLMNATSHR
SCHEMBL5225071 0.78 CASR (0.51) MAPTLMNATSHRHTT
SCHEMBL5217387 0.77 CASR (0.41) ALDH1A1MAPTLMNATSHRHTT
SCHEMBL23704670 0.77 LMNA (0.40) ALDH1A1MAPTLMNATSHRHTT
SCHEMBL17427512 0.76 HTR1B (0.40) ALDH1A1KDM4EMAPTLMNATSHR
SCHEMBL1154287 0.76 MCL1 (0.55) ALDH1A1KDM4EMAPTLMNAHTT
SCHEMBL5217886 0.75 HRH1 (0.41) ALDH1A1KDM4EMAPTLMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765810-A1 2,4-DIAMINOQUINAZOLINES FOR SPINAL MUSCULAR ATROPHY Decode Chemistry, Inc. (US) 2007-03-28 EP disclosed
WO-2005123724-A1 2,4-DIAMINOQUINAZOLINES FOR SPINAL MUSCULAR ATROPHY DECODE CHEMISTRY, INC. (US) 2005-12-29 WO disclosed