SCHEMBL5223526

SCHEMBL5223526

N#Cc1c(F)cccc1OCCc1ccccc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 6/20 0.43
KCNH2 Q12809 2/20 0.41
CASR P41180 2/20 0.40
LMNA P02545 2/20 0.40
MAPT P10636 2/20 0.40
TSHR P16473 2/20 0.40
HTT P42858 2/20 0.40
TAAR1 Q96RJ0 1/20 0.39
MRGPRX4 Q96LA9 1/20 0.38
BRD4 O60885 1/20 0.37
POLB P06746 1/20 0.37
HPGD P15428 1/20 0.37
MAPK1 P28482 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
NRP1 O14786 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
P2RX7 Q99572 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5217402 0.89 LMNA (0.43) LMNAMAPTTSHRHTTTAAR1
SCHEMBL1154503 0.86 HSD11B1 (0.50) HSD11B1LMNAMAPTTSHRHTT
SCHEMBL5219882 0.83 ALDH1A1 (0.46) LMNAMAPTTSHRHTTHPGD
SCHEMBL1154474 0.80 CYP11B1 (0.43) LMNAMAPTTSHRHTTMRGPRX4
SCHEMBL5216704 0.80 MAPT (0.42) CASRLMNAMAPTTSHRHTT
SCHEMBL1155054 0.80 NPC1 (0.52) CASRLMNAMAPTTSHRHTT
SCHEMBL5221531 0.79 CASR (0.41) KCNH2CASRLMNAMAPTTSHR
SCHEMBL5217387 0.79 CASR (0.41) KCNH2CASRLMNAMAPTTSHR
SCHEMBL23704670 0.78 LMNA (0.40) LMNAMAPTTSHRHTTTAAR1
SCHEMBL2164306 0.78 HSD11B1 (0.41) HSD11B1CASRP2RX7MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765810-A1 2,4-DIAMINOQUINAZOLINES FOR SPINAL MUSCULAR ATROPHY Decode Chemistry, Inc. (US) 2007-03-28 EP disclosed
WO-2005123724-A1 2,4-DIAMINOQUINAZOLINES FOR SPINAL MUSCULAR ATROPHY DECODE CHEMISTRY, INC. (US) 2005-12-29 WO disclosed