SCHEMBL5220117

SCHEMBL5220117

CCn1ccc2c(N3CCCS3(O)O)cc(C(=O)O)cc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.37
CTSD P07339 1/20 0.37
BACE2 Q9Y5Z0 1/20 0.37
CYP19A1 P11511 1/20 0.33
DRD3 P35462 1/20 0.33
POLB P06746 2/20 0.32
RHEB Q15382 1/20 0.31
KDM4E B2RXH2 4/20 0.31
ALDH1A1 P00352 4/20 0.31
HPGD P15428 4/20 0.31
HSD17B10 Q99714 3/20 0.31
SLC22A12 Q96S37 2/20 0.31
TSHR P16473 2/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
KMT2A Q03164 1/20 0.31
BRD4 O60885 1/20 0.30
LMNA P02545 1/20 0.30
HTT P42858 1/20 0.30
CYP2J2 P51589 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5218348 0.97 BACE1 (0.37) BACE1CTSDBACE2CYP19A1DRD3
SCHEMBL5220119 0.89 POLB (0.42) BACE1CTSDBACE2CYP19A1DRD3
SCHEMBL5220034 0.88 BACE1 (0.37) BACE1CTSDBACE2POLBKDM4E
SCHEMBL5218338 0.85 POLB (0.46) BACE1CTSDBACE2CYP19A1DRD3
SCHEMBL5222272 0.85 BACE1 (0.37) BACE1CTSDBACE2POLBKDM4E
SCHEMBL5222586 0.79 CTSD (0.37) BACE1CTSDBACE2KDM4EALDH1A1
SCHEMBL5225090 0.77 BACE1 (0.53) BACE1CTSDBACE2KDM4EALDH1A1
SCHEMBL5217639 0.76 CTSD (0.37) BACE1CTSDBACE2POLBHPGD
SCHEMBL308351 0.75 NPC1 (0.44) POLBKDM4EALDH1A1HPGDHSD17B10
SCHEMBL5219142 0.74 BACE1 (0.58) BACE1CTSDBACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed