SCHEMBL5220505

SCHEMBL5220505

O=[N+]([O-])c1cccc(-c2ccc(C34CCCN(CC3)C4)cn2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42
IDO1 P14902 1/20 0.41
KMT2A Q03164 1/20 0.41
MAPT P10636 5/20 0.40
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
ALDH1A1 P00352 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
CYP1A2 P05177 1/20 0.39
KEAP1 Q14145 2/20 0.38
NFE2L2 Q16236 2/20 0.38
ECE1 P42892 1/20 0.38
MET P08581 1/20 0.38
PGR P06401 1/20 0.38
PLK1 P53350 1/20 0.38
LMNA P02545 1/20 0.38
THRB P10828 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CASP3 P42574 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL4472025 0.99 RAB9A (0.41) RAB9ANPC1IDO1KMT2AMAPT
SCHEMBL4466231 0.81 HPGDS (0.41) IDO1BCHEACHE
SCHEMBL5156396 0.81 KDM1A (0.43) IDO1KMT2A
SCHEMBL4473786 0.81 RAB9A (0.40) RAB9ANPC1IDO1KMT2AMAPT
SCHEMBL4463296 0.80 HSD11B1 (0.40)
Bromide SCHEMBL4466442 0.80 KDM1A (0.42) IDO1KMT2A
Bromide SCHEMBL4480660 0.80 HPGDS (0.41) IDO1
Bromide SCHEMBL4471147 0.79 HSD11B1 (0.39)
SCHEMBL2678219 0.78 HPGDS (0.43) IDO1BCHEACHE
SCHEMBL2678305 0.78 KDM1A (0.47) RAB9ANPC1KMT2AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465893-B1 DERIVATIVES OF 5-(PYRIDIN-3-YL)-1-AZABICYCLO (3.2.1) OCTANE, THE PREPARATION THEREOF AND THE APPLICATION OF SAME IN THERAPEUTICS SANOFI AVENTIS (FR) 2007-02-28 EP claimed