SCHEMBL5220548

SCHEMBL5220548

CC(C)(C)N(C(=O)O)[C@@H](Cc1ccccc1Cl)[C@@H](O)CNC1CCCCC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.44
LMNA P02545 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
SCN1A P35498 1/20 0.42
SCN2A Q99250 1/20 0.42
SCN3A Q9NY46 1/20 0.42
BACE1 P56817 2/20 0.39
CTSD P07339 1/20 0.39
BACE2 Q9Y5Z0 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
POLB P06746 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 2/20 0.37
ALDH1A1 P00352 2/20 0.37
ALOX15 P16050 1/20 0.37
SLC16A3 O15427 1/20 0.36
SLC16A1 P53985 1/20 0.36
MCTS1 Q9ULC4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5220541 1.00 KDM4E (0.44) KDM4ELMNACYP1A2CYP2D6SCN1A
SCHEMBL5218781 0.83 POLB (0.43) KDM4ELMNACYP1A2CYP2D6SCN1A
SCHEMBL5218771 0.83 POLB (0.43) KDM4ELMNACYP1A2CYP2D6SCN1A
SCHEMBL5224070 0.82 EPHX2 (0.47) KDM4ELMNACYP1A2CYP2D6BACE1
SCHEMBL5224084 0.82 EPHX2 (0.47) KDM4ELMNACYP1A2CYP2D6BACE1
SCHEMBL5221255 0.80 USP2 (0.46) KDM4ELMNACYP1A2CYP2D6SCN1A
SCHEMBL5221262 0.80 USP2 (0.46) KDM4ELMNACYP1A2CYP2D6SCN1A
SCHEMBL4693111 0.76 BACE1 (0.41) BACE1CTSDBACE2
SCHEMBL5223476 0.76 BACE1 (0.44) BACE1CTSDBACE2
SCHEMBL5223435 0.76 BACE1 (0.42) BACE1CTSDBACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed