SCHEMBL5221262

SCHEMBL5221262

CC(C)(C)N(C(=O)O)[C@@H](Cc1ccco1)[C@@H](O)CNC1CCCCC1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.46
TSHR P16473 4/20 0.45
ALDH1A1 P00352 3/20 0.45
LMNA P02545 2/20 0.45
NPSR1 Q6W5P4 2/20 0.45
KDM4E B2RXH2 1/20 0.42
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
SCN1A P35498 1/20 0.40
SCN2A Q99250 1/20 0.40
SCN3A Q9NY46 1/20 0.40
HPGD P15428 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TP53 P04637 1/20 0.39
MAPK1 P28482 1/20 0.39
CTSD P07339 1/20 0.38
BACE1 P56817 1/20 0.38
BACE2 Q9Y5Z0 1/20 0.38
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5221255 1.00 USP2 (0.46) USP2TSHRALDH1A1LMNANPSR1
SCHEMBL5220541 0.80 KDM4E (0.44) TSHRALDH1A1LMNANPSR1KDM4E
SCHEMBL5220548 0.80 KDM4E (0.44) TSHRALDH1A1LMNANPSR1KDM4E
SCHEMBL5218771 0.80 POLB (0.43) LMNAKDM4ECYP1A2CYP2D6SCN1A
SCHEMBL5218781 0.80 POLB (0.43) LMNAKDM4ECYP1A2CYP2D6SCN1A
SCHEMBL5223196 0.79 CTSD (0.38) TSHRALDH1A1NPSR1MAPK1CTSD
SCHEMBL5224070 0.79 EPHX2 (0.47) TSHRALDH1A1LMNAKDM4ECYP1A2
SCHEMBL5223208 0.79 CTSD (0.38) TSHRALDH1A1NPSR1MAPK1CTSD
SCHEMBL5224084 0.79 EPHX2 (0.47) TSHRALDH1A1LMNAKDM4ECYP1A2
SCHEMBL4693114 0.77 BACE1 (0.41) CTSDBACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed