SCHEMBL5221564

SCHEMBL5221564

CCn1nnc2c(N3CCCC3=O)cc(C(=O)O)cc21

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSD P07339 3/20 0.51
BACE1 P56817 3/20 0.51
BACE2 Q9Y5Z0 3/20 0.51
HCAR3 P49019 4/20 0.44
ALDH1A1 P00352 2/20 0.40
CYP2C9 P11712 4/20 0.40
CYP3A4 P08684 2/20 0.40
HPGD P15428 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
GAA P10253 1/20 0.36
HSD17B10 Q99714 1/20 0.36
RARA P10276 1/20 0.34
RARB P10826 1/20 0.34
RARG P13631 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
USP2 O75604 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5216173 0.90 CTSD (0.49) CTSDBACE1BACE2HCAR3ALDH1A1
SCHEMBL5219279 0.79 CTSD (0.51) CTSDBACE1BACE2ALDH1A1CYP2C9
SCHEMBL5220770 0.79 BACE1 (0.52) CTSDBACE1BACE2ALDH1A1CYP2C9
SCHEMBL5216179 0.76 MAPT (0.44) CTSDBACE1BACE2ALDH1A1CYP2C9
SCHEMBL5225090 0.73 BACE1 (0.53) CTSDBACE1BACE2ALDH1A1CYP2C9
SCHEMBL5221894 0.70 BACE1 (0.49) CTSDBACE1BACE2ALDH1A1CYP2C9
SCHEMBL5218022 0.70 BACE1 (0.50) CTSDBACE1BACE2ALDH1A1CYP2C9
SCHEMBL5217707 0.70 ALDH1A1 (0.54) ALDH1A1CYP2C9CYP3A4HPGDCYP1A2
SCHEMBL5222262 0.69 ALDH1A1 (0.50) ALDH1A1CYP2C9CYP3A4HPGDCYP1A2
SCHEMBL5219489 0.68 ALDH1A1 (0.47) CTSDBACE1BACE2ALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed