SCHEMBL5222341

SCHEMBL5222341

COc1ccccc1C(C)Oc1cccc(F)c1C#N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.41
DRD2 P14416 1/20 0.41
HRH1 P35367 1/20 0.41
ALDH1A1 P00352 2/20 0.39
SQOR Q9Y6N5 2/20 0.37
NFE2L2 Q16236 1/20 0.36
ADRA2A P08913 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
AR P10275 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
IKBKE Q14164 2/20 0.35
HIF1A Q16665 1/20 0.35
SLC6A4 P31645 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1155267 0.91 ALDH1A1 (0.41) HTR2ADRD2HRH1ALDH1A1ADRA2A
SCHEMBL1155296 0.86 IKBKE (0.39) HTR2ADRD2HRH1ALDH1A1ADRA2A
SCHEMBL1155272 0.85 ALDH1A1 (0.37) HTR2ADRD2HRH1ALDH1A1SQOR
SCHEMBL1155211 0.85 ALDH1A1 (0.37) HTR2ADRD2HRH1ALDH1A1SQOR
SCHEMBL1154973 0.85 ALDH1A1 (0.37) HTR2ADRD2HRH1ALDH1A1SQOR
SCHEMBL1154756 0.84 IKBKE (0.43) HTR2ADRD2HRH1ALDH1A1ADRA2A
SCHEMBL1155086 0.82 HTR6 (0.40) HTR2ADRD2HRH1ALDH1A1ADRA2A
SCHEMBL1154472 0.82 HTR6 (0.40) HTR2ADRD2HRH1ALDH1A1ADRA2A
SCHEMBL1155061 0.82 HTR6 (0.40) HTR2ADRD2HRH1ALDH1A1ADRA2A
SCHEMBL1155196 0.82 DRD2 (0.39) HTR2ADRD2HRH1ALDH1A1ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765810-A1 2,4-DIAMINOQUINAZOLINES FOR SPINAL MUSCULAR ATROPHY Decode Chemistry, Inc. (US) 2007-03-28 EP disclosed
WO-2005123724-A1 2,4-DIAMINOQUINAZOLINES FOR SPINAL MUSCULAR ATROPHY DECODE CHEMISTRY, INC. (US) 2005-12-29 WO disclosed