SCHEMBL5222480

SCHEMBL5222480

CCNc1cc(C(=O)OC)cc(N2CCCS2(=O)=O)c1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 2/20 0.44
BACE1 P56817 2/20 0.44
BACE2 Q9Y5Z0 2/20 0.44
PIK3C3 Q8NEB9 2/20 0.39
TP53 P04637 7/20 0.39
RPS6KB1 P23443 1/20 0.38
AKT1 P31749 1/20 0.38
MAPT P10636 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
ALDH1A1 P00352 3/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
TSHR P16473 1/20 0.36
KDM4E B2RXH2 2/20 0.35
LMNA P02545 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4D Q08499 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5218030 0.97 BACE1 (0.47) CTSDBACE1BACE2PIK3C3TP53
SCHEMBL5222633 0.89 CTSD (0.48) CTSDBACE1BACE2PIK3C3TP53
SCHEMBL5219825 0.88 BACE1 (0.47) CTSDBACE1BACE2PIK3C3TP53
SCHEMBL5218025 0.86 BACE1 (0.41) CTSDBACE1BACE2RPS6KB1AKT1
SCHEMBL5218051 0.85 BACE1 (0.51) CTSDBACE1BACE2TP53SMN1; SMN2
SCHEMBL5219490 0.85 BACE1 (0.50) CTSDBACE1BACE2PIK3C3TP53
SCHEMBL5219375 0.82 KDM4E (0.48) PIK3C3TP53MAPTSMN1; SMN2ALDH1A1
SCHEMBL5218053 0.80 CTSD (0.49) CTSDBACE1BACE2PIK3C3TP53
SCHEMBL5219941 0.79 POLB (0.37) CTSDBACE1BACE2PIK3C3TP53
SCHEMBL5219776 0.79 KDM4E (0.50) PIK3C3TP53MAPTSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed