SCHEMBL5222633

SCHEMBL5222633

CCNc1cc(C(=O)OC)cc(N2CCCS2(=O)=O)c1OC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 3/20 0.48
BACE1 P56817 3/20 0.48
BACE2 Q9Y5Z0 3/20 0.48
PDE4B Q07343 1/20 0.38
PDE4D Q08499 1/20 0.38
TP53 P04637 5/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
PIK3C3 Q8NEB9 2/20 0.36
MAPT P10636 1/20 0.36
POLB P06746 1/20 0.35
ALDH1A1 P00352 5/20 0.35
TSHR P16473 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
KDM4E B2RXH2 4/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
GAA P10253 1/20 0.33
ALOX15 P16050 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5218051 0.97 BACE1 (0.51) CTSDBACE1BACE2PDE4BPDE4D
SCHEMBL5218053 0.91 CTSD (0.49) CTSDBACE1BACE2PDE4BPDE4D
SCHEMBL5222641 0.89 CTSD (0.41) CTSDBACE1BACE2PDE4BPDE4D
SCHEMBL5222480 0.89 CTSD (0.44) CTSDBACE1BACE2PDE4BPDE4D
SCHEMBL5220748 0.88 BACE1 (0.52) CTSDBACE1BACE2PDE4BPDE4D
SCHEMBL5218055 0.86 CTSD (0.44) CTSDBACE1BACE2PDE4BPDE4D
SCHEMBL5218030 0.85 BACE1 (0.47) CTSDBACE1BACE2TP53SMN1; SMN2
SCHEMBL5220487 0.81 KDM4E (0.47) TP53SMN1; SMN2PIK3C3MAPTPOLB
SCHEMBL5218045 0.80 CTSD (0.42) CTSDBACE1BACE2PDE4BPDE4D
SCHEMBL5221138 0.78 KDM4E (0.49) CTSDBACE1BACE2TP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed