SCHEMBL5222786

SCHEMBL5222786

CN(C)C1CCN(Cc2cnn(-c3ccc(-c4ccc(F)cc4)cc3)c2-c2ccco2)C1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.38
MCHR1 Q99705 2/20 0.36
KDM1A O60341 1/20 0.36
SMO Q99835 1/20 0.35
PTGS1 P23219 1/20 0.34
MAP4K4 O95819 2/20 0.34
CXCR3 P49682 1/20 0.34
CYP2D6 P10635 1/20 0.33
HRH1 P35367 1/20 0.33
KCNH2 Q12809 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MITF O75030 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TP53 P04637 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
LTA4H P09960 1/20 0.33
PLA2G7 Q13093 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5225875 0.85 CYP2D6 (0.36) KDM1ASMOPTGS1CXCR3CYP2D6
SCHEMBL5228002 0.83 TSHR (0.39) MCHR1SMOPTGS1KDM4ETP53
SCHEMBL2761237 0.82 SMO (0.43) SMOPTGS1KDM4EL3MBTL1TP53
SCHEMBL2761009 0.82 SMO (0.43) SMOPTGS1L3MBTL1TP53SMN1; SMN2
SCHEMBL5224732 0.81 MAP4K4 (0.34) MCHR1PTGS1MAP4K4CYP2D6HRH1
Hydrochloric Acid SCHEMBL1997589 0.81 SMO (0.42) SMOPTGS1KDM4EL3MBTL1TP53
SCHEMBL2761177 0.80 DRD4 (0.42) SMOPTGS1KDM4ETP53
SCHEMBL2761137 0.80 SMO (0.41) SMOPTGS1L3MBTL1TP53SMN1; SMN2
SCHEMBL5223970 0.79 ADORA2A (0.40) MCHR1SMOPTGS1KCNH2L3MBTL1
SCHEMBL5228047 0.79 HTR2C (0.37) MCHR1CXCR3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed