SCHEMBL5225875

SCHEMBL5225875

OCC1CCN(Cc2cnn(-c3ccc(-c4ccc(F)cc4)cc3)c2-c2ccco2)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.36
PTGS1 P23219 1/20 0.34
SMO Q99835 1/20 0.34
CCR3 P51677 1/20 0.34
NR3C1 P04150 2/20 0.33
POLB P06746 2/20 0.33
CXCR3 P49682 1/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
CYP3A4 P08684 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ALDH1A1 P00352 1/20 0.32
KDM1A O60341 1/20 0.32
TP53 P04637 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
DRD2 P14416 1/20 0.32
DRD4 P21917 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5228002 0.85 TSHR (0.39) PTGS1SMOPOLBALDH1A1TP53
SCHEMBL5222786 0.85 GRM2 (0.38) CYP2D6PTGS1SMOCXCR3KDM1A
SCHEMBL5228047 0.81 HTR2C (0.37) CXCR3ALDH1A1DRD2DRD4
SCHEMBL2761237 0.81 SMO (0.43) PTGS1SMOMAPTALDH1A1TP53
SCHEMBL2761009 0.81 SMO (0.43) PTGS1SMOMAPTALDH1A1TP53
SCHEMBL2761177 0.81 DRD4 (0.42) PTGS1SMOPOLBMAPTALDH1A1
SCHEMBL5225031 0.81 SSTR5 (0.36) CYP2D6SMO
SCHEMBL2001019 0.81 CXCR3 (0.36) CXCR3
SCHEMBL2000116 0.81 F10 (0.38) NR3C1PDCD1CD274
Hydrochloric Acid SCHEMBL1997589 0.80 SMO (0.42) PTGS1SMOMAPTALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed