SCHEMBL5228047

SCHEMBL5228047

OC1CCN(Cc2cnn(-c3ccc(-c4cccc(F)c4)cc3)c2-c2ccco2)C1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.37
MCHR1 Q99705 2/20 0.37
DRD2 P14416 1/20 0.37
DRD4 P21917 1/20 0.37
ALDH1A1 P00352 2/20 0.36
ALPL P05186 1/20 0.36
KDM4E B2RXH2 1/20 0.36
HTT P42858 1/20 0.36
ADRB2 P07550 2/20 0.36
ROCK2 O75116 2/20 0.36
GAA P10253 1/20 0.35
CXCR3 P49682 1/20 0.34
F10 P00742 3/20 0.34
DHODH Q02127 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5229287 0.88 EGFR (0.40) ALDH1A1ALPLKDM4EHTTGAA
SCHEMBL5228002 0.87 TSHR (0.39) HTR2CMCHR1ALDH1A1KDM4EHTT
SCHEMBL5226446 0.86 ALDH1A1 (0.41) ALDH1A1KDM4EGAA
SCHEMBL5227634 0.85 PDCD1 (0.40) ALDH1A1KDM4E
SCHEMBL1998836 0.84 HTR2C (0.39) HTR2CMCHR1CXCR3F10ADORA2A
SCHEMBL2003024 0.84 HTR2C (0.37) HTR2CMCHR1ALDH1A1ROCK2GAA
SCHEMBL5228505 0.84 F10 (0.48) F10
SCHEMBL5224673 0.84 SMO (0.40) DRD2DRD4ALDH1A1ALPLKDM4E
SCHEMBL5224744 0.84 HTR1A (0.38) HTR2CALDH1A1ALPLKDM4EROCK2
SCHEMBL5226613 0.84 SMO (0.40) DRD2DRD4ALDH1A1ALPLKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed