SCHEMBL5224099

SCHEMBL5224099

Cn1c(N(C(=O)O)c2ccc(C(C)(C)C)cc2)nc2cc(N)ccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GCGR P47871 2/20 0.38
HDAC6 Q9UBN7 3/20 0.38
NPC1 O15118 2/20 0.37
GFER P55789 2/20 0.37
RAB9A P51151 1/20 0.37
KDM4E B2RXH2 4/20 0.34
HTT P42858 2/20 0.34
EPHX2 P34913 1/20 0.34
NR1H4 Q96RI1 1/20 0.34
BRAF P15056 2/20 0.34
RAF1 P04049 1/20 0.34
NPC1L1 Q9UHC9 1/20 0.34
ALDH1A1 P00352 3/20 0.34
TDP1 Q9NUW8 3/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
GCG P01275 1/20 0.33
GIPR P48546 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5230034 0.87 NPC1 (0.40) HDAC6NPC1GFERRAB9AKDM4E
SCHEMBL4978649 0.87 BRD4 (0.35) GCGRHDAC6NPC1GFERRAB9A
SCHEMBL5226357 0.87 HDAC6 (0.48) HDAC6NPC1GFERRAB9AKDM4E
SCHEMBL5226340 0.86 HDAC6 (0.39) GCGRHDAC6NPC1GFERRAB9A
SCHEMBL5222469 0.84 ALDH1A1 (0.44) HDAC6NPC1RAB9AKDM4EALDH1A1
SCHEMBL4980289 0.78 HDAC6 (0.41) HDAC6NPC1RAB9AKDM4ENPC1L1
SCHEMBL5226042 0.77 KDR (0.37) GCGRHDAC6BRAFRAF1HDAC3
SCHEMBL4978515 0.77 BRD4 (0.38) GCGRHDAC6NPC1GFERRAB9A
SCHEMBL5226236 0.77 BRAF (0.45) GCGRHDAC6NPC1RAB9AKDM4E
SCHEMBL4978242 0.76 BRD4 (0.35) GCGRHDAC6NPC1GFERRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487824-B1 DIAMINO-PYRIMIDINES AND THEIR USE AS ANGIOGENESIS INHIBITORS SMITHKLINE BEECHAM CORP (US) 2007-06-20 EP disclosed