SCHEMBL5222469

SCHEMBL5222469

COc1ccc(N(C(=O)O)c2nc3cc(N)ccc3n2C)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
MAPT P10636 2/20 0.44
ACSS2 Q9NR19 1/20 0.39
KDM4E B2RXH2 4/20 0.39
HSD17B10 Q99714 2/20 0.39
HPGD P15428 2/20 0.39
TDP1 Q9NUW8 1/20 0.38
F2 P00734 1/20 0.38
HDAC6 Q9UBN7 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
GAA P10253 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
ITK Q08881 1/20 0.37
FGFR1 P11362 1/20 0.37
BTK Q06187 1/20 0.37
HDAC1 Q13547 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5230034 0.87 NPC1 (0.40) ALDH1A1SMN1; SMN2MAPTACSS2KDM4E
SCHEMBL5226357 0.87 HDAC6 (0.48) ALDH1A1MAPTKDM4EHSD17B10HPGD
SCHEMBL4982539 0.86 ALDH1A1 (0.42) ALDH1A1SMN1; SMN2MAPTACSS2KDM4E
SCHEMBL5226340 0.86 HDAC6 (0.39) ALDH1A1SMN1; SMN2MAPTKDM4EHSD17B10
SCHEMBL5224099 0.84 GCGR (0.38) ALDH1A1MAPTKDM4EHSD17B10HPGD
SCHEMBL5226510 0.83 MAPT (0.54) ALDH1A1SMN1; SMN2MAPTKDM4ENPC1
SCHEMBL5224606 0.77 KDR (0.37) ALDH1A1SMN1; SMN2ACSS2KDM4EHSD17B10
SCHEMBL5230055 0.77 BRAF (0.39) ALDH1A1SMN1; SMN2MAPTKDM4EHSD17B10
SCHEMBL14274200 0.76 HDAC6 (0.41) ALDH1A1MAPTKDM4EHSD17B10HPGD
SCHEMBL4980289 0.76 HDAC6 (0.41) ALDH1A1ACSS2KDM4EF2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487824-B1 DIAMINO-PYRIMIDINES AND THEIR USE AS ANGIOGENESIS INHIBITORS SMITHKLINE BEECHAM CORP (US) 2007-06-20 EP disclosed