SCHEMBL5226340

SCHEMBL5226340

Cn1c(N(C(=O)O)c2ccc(F)cc2)nc2cc(N)ccc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 4/20 0.39
F2 P00734 1/20 0.38
KDM4E B2RXH2 4/20 0.36
ALDH1A1 P00352 3/20 0.36
HPGD P15428 2/20 0.36
HSD17B10 Q99714 2/20 0.36
HDAC3 O15379 1/20 0.36
PTGS1 P23219 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
TDP1 Q9NUW8 2/20 0.36
NPC1 O15118 5/20 0.35
MAPT P10636 2/20 0.35
HTT P42858 2/20 0.35
POLB P06746 1/20 0.35
GFER P55789 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5230034 0.89 NPC1 (0.40) HDAC6KDM4EALDH1A1HPGDHSD17B10
SCHEMBL5226357 0.89 HDAC6 (0.48) HDAC6F2KDM4EALDH1A1HPGD
SCHEMBL5224099 0.86 GCGR (0.38) HDAC6F2KDM4EALDH1A1HPGD
SCHEMBL5222469 0.86 ALDH1A1 (0.44) HDAC6F2KDM4EALDH1A1HPGD
SCHEMBL4978242 0.85 BRD4 (0.35) HDAC6F2KDM4EALDH1A1HPGD
SCHEMBL5224254 0.76 KDR (0.38) HDAC6F2HDAC3PTGS1HDAC4
SCHEMBL5226590 0.76 GRM5 (0.38) HDAC6ALDH1A1HSD17B10NPC1MAPT
SCHEMBL14274200 0.75 HDAC6 (0.41) HDAC6F2KDM4EALDH1A1HPGD
SCHEMBL4980289 0.75 HDAC6 (0.41) HDAC6F2KDM4EALDH1A1HDAC1
SCHEMBL4978515 0.74 BRD4 (0.38) HDAC6KDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487824-B1 DIAMINO-PYRIMIDINES AND THEIR USE AS ANGIOGENESIS INHIBITORS SMITHKLINE BEECHAM CORP (US) 2007-06-20 EP disclosed