SCHEMBL5224710

SCHEMBL5224710

Nc1cccc(NC(=O)OC(c2ccncc2)C2CCNCC2)c1N

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 11/20 0.44
SLC6A2 P23975 9/20 0.44
SLC6A3 Q01959 6/20 0.44
CYP2D6 P10635 1/20 0.36
KCNH2 Q12809 1/20 0.36
SMYD3 Q9H7B4 1/20 0.35
CHRM3 P20309 1/20 0.35
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7244377 0.82 SLC6A4 (0.44) SLC6A4SLC6A2SLC6A3
Hydrochloric Acid SCHEMBL5228421 0.77 MEN1 (0.45) SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL5225301 0.77 RAB9A (0.54) HDAC3HDAC1HDAC2
Hydrochloric Acid SCHEMBL5227582 0.75 AKT1 (0.46) SLC6A4SLC6A2SLC6A3
SCHEMBL5224189 0.74 SLC6A4 (0.44) SLC6A4SLC6A2SLC6A3
SCHEMBL5225038 0.73 GPR132 (0.48) HDAC1
SCHEMBL27747825 0.73 SLC6A4 (0.50) SLC6A4SLC6A2SLC6A3
SCHEMBL7380676 0.70 SLC6A4 (0.66) SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL5226962 0.70 CYP17A1 (0.36) SLC6A4SLC6A2SLC6A3
SCHEMBL7244090 0.68 CYP17A1 (0.36) SLC6A4SLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1014962-A4 ANTITHROMBOTIC AGENTS LILLY CO ELI (US) 2007-06-27 EP disclosed
EP-1014962-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 2000-07-05 EP disclosed
WO-1999000121-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 1999-01-07 WO disclosed